WIPO logo
Mobile | Deutsch | Español | Français | 日本語 | 한국어 | Português | Русский | 中文 | العربية |
PATENTSCOPE

Search International and National Patent Collections
World Intellectual Property Organization
Search
 
Browse
 
Translate
 
Options
 
News
 
Login
 
Help
 
Machine translation
1. (WO2012110774) SELECTIVE FAK INHIBITORS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2012/110774    International Application No.:    PCT/GB2012/000176
Publication Date: 23.08.2012 International Filing Date: 17.02.2012
IPC:
C07D 239/42 (2006.01), C07D 401/12 (2006.01), A61K 31/506 (2006.01), A61P 35/00 (2006.01)
Applicants: CANCER THERAPEUTICS CRC PTY LIMITED [AU/AU]; 4 Research Avenu Bundoora, VIC 3083 (AU) (For All Designated States Except US).
HOLMES, Ian, Peter [GB/AU]; (AU) (For US Only).
BERGMAN, Ylva [SE/AU]; (AU) (For US Only).
LUNNISS, Gillian Elizabeth [GB/AU]; (AU) (For US Only).
NIKAC, Marica [AU/AU]; (AU) (For US Only).
CHOI, Neil [AU/AU]; (AU) (For US Only).
HEMLEY, Catherine Fae [AU/AU]; (AU) (For US Only).
WALKER, Scott Raymond [NZ/AU]; (AU) (For US Only).
FOITZIK, Richard Charles [AU/AU]; (AU) (For US Only).
GANAME, Danny [AU/AU]; (AU) (For US Only).
LESSENE, Romina [AU/AU]; (AU) (For US Only)
Inventors: HOLMES, Ian, Peter; (AU).
BERGMAN, Ylva; (AU).
LUNNISS, Gillian Elizabeth; (AU).
NIKAC, Marica; (AU).
CHOI, Neil; (AU).
HEMLEY, Catherine Fae; (AU).
WALKER, Scott Raymond; (AU).
FOITZIK, Richard Charles; (AU).
GANAME, Danny; (AU).
LESSENE, Romina; (AU)
Agent: WATSON, Robert James; Mewburn Ellis LLP 33 Gutter Lane London EC2V 8AS (GB)
Priority Data:
61/443,773 17.02.2011 US
61/523,489 15.08.2011 US
61/579,729 23.12.2011 US
Title (EN) SELECTIVE FAK INHIBITORS
(FR) INHIBITEURS SÉLECTIFS DE FAK
Abstract: front page image
(EN)A compound of the formula (I) where R1 or R2 is a cycle amine group and R5 is an aromatic group with a carbonyl containing substituent for use as a FAK inhibitor.
(FR)La présente invention concerne un composé de formule (I), dans laquelle R1 ou R2 est un groupe amine cyclique et R5 est un groupe aromatique avec un substituant contenant un carbonyle destiné à être utilisé en tant qu'inhibiteur de FAK.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)