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1. (WO2012103279) METHODS AND COMPOSITIONS FOR THE SYNTHESIS OF MULTIMERIZING AGENTS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2012/103279    International Application No.:    PCT/US2012/022642
Publication Date: 02.08.2012 International Filing Date: 26.01.2012
IPC:
C07D 319/06 (2006.01)
Applicants: ARIAD PHARMACEUTICALS, INCORPORATED [US/US]; 26 Landsdowne Street Cambridge, MA 02139 (US) (For All Designated States Except US).
LI, Feng [CN/US]; (US) (For US Only).
WANG, Yihan [CN/US]; (US) (For US Only)
Inventors: LI, Feng; (US).
WANG, Yihan; (US)
Agent: ELLISON, Jeffrey J.; Clark & Elbing LLP 101 Federal Street Boston, MA 02110 (US)
Priority Data:
61/436,430 26.01.2011 US
Title (EN) METHODS AND COMPOSITIONS FOR THE SYNTHESIS OF MULTIMERIZING AGENTS
(FR) PROCÉDÉS ET COMPOSITIONS POUR LA SYNTHÈSE D'AGENTS DE MULTIMÉRISATION
Abstract: front page image
(EN)The invention features methods and compositions for the synthesis of multimerizing agents. An exemplary method for producing AP20187 may comprise: (a) coupling 2-N,Ndimethylaminomethyl-1,3-diaminopropane with AP20792 to produce the dimeric alcohol, AP20793; and (b) coupling the AP20793 so produced with API7362 to yield AP20187. In particular embodiments, the method further includes the step of producing API7362 by coupling API7360 with methyl-L-pipecolic acid, or a salt thereof.
(FR)Procédés et compositions pour la synthèse d'agents de multimérisation.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)