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1. (WO2012097000) PROCESSES FOR PREPARING ISOQUINOLINONES AND SOLID FORMS OF ISOQUINOLINONES
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2012/097000 International Application No.: PCT/US2012/020831
Publication Date: 19.07.2012 International Filing Date: 10.01.2012
IPC:
A61K 31/497 (2006.01)
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
495
having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
4965
Non-condensed pyrazines
497
containing further heterocyclic rings
Applicants:
INFINITY PHARMACEUTICALS, INC. [US/US]; 780 Memorial Drive Cambridge, MA 02139, US (AllExceptUS)
INTELLIKINE LLC [US/US]; 10931 N. Torrey Pines Road Suite 103 La Jolla, CA 92037, US (AllExceptUS)
REN, Pingda [CN/US]; US (UsOnly)
MARTIN, Michael [US/US]; US (UsOnly)
ISBESTER, Paul [US/US]; US (UsOnly)
LANE, Benjamin, S. [US/US]; US (UsOnly)
KROPP, Jason [US/US]; US (UsOnly)
Inventors:
REN, Pingda; US
MARTIN, Michael; US
ISBESTER, Paul; US
LANE, Benjamin, S.; US
KROPP, Jason; US
Agent:
MCCARTY, Catherine, M.; Lando & Anastasi LLP Riverfront Office Park One Main Street, Suite 1100 Cambridge, MA 02142, US
Priority Data:
61/431,30410.01.2011US
61/578,65521.12.2011US
Title (EN) PROCESSES FOR PREPARING ISOQUINOLINONES AND SOLID FORMS OF ISOQUINOLINONES
(FR) PROCÉDÉS DE PRÉPARATION D'ISOQUINOLINONES ET DE FORMES SOLIDES D'ISOQUINOLINONES
Abstract:
(EN) Polymorphs of chemical compounds that modulate kinase activity, including PI3 kinase activity, and compounds, pharmaceutical compositions, and methods of treatment of diseases and conditions associated with kinase activity, including PI 3 kinase activity, are described herein. Also provided herein are processes for preparing compounds, polymorphs thereof, and pharmaceutical compositions thereof.
(FR) La présente invention a pour objet des polymorphes de composés chimiques qui modulent l'activité de la kinase, y compris l'activité de la PI3 kinase, et des composés, des compositions pharmaceutiques, et des méthodes de traitement de maladies et d'affections associées à l'activité de la kinase, y compris l'activité de la PI 3 kinase. La présente invention concerne également des procédés de préparation des composés, de leurs polymorphes, et de leurs compositions pharmaceutiques.
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Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)
Also published as:
UAa201309964CA2824197EP2663309JP2014501790SG191897RU2013137424
KR1020140020249NZ612909AU2012205669RU0002626883MYPI 2013701203PH1/2013/501465
ES2637113EP3238722IL227387KR1020180080358PH1/2018/500960