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1. (WO2012053186) ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2012/053186    International Application No.:    PCT/JP2011/005802
Publication Date: 26.04.2012 International Filing Date: 18.10.2011
Chapter 2 Demand Filed:    20.08.2012    
IPC:
C07D 213/81 (2006.01), A61K 31/44 (2006.01), A61K 31/4427 (2006.01), A61K 31/444 (2006.01), A61K 31/506 (2006.01), A61P 25/00 (2006.01), A61P 29/00 (2006.01), A61P 43/00 (2006.01), C07D 213/64 (2006.01), C07D 239/42 (2006.01), C07D 401/04 (2006.01), C07D 401/12 (2006.01), C07D 401/14 (2006.01), C07D 405/12 (2006.01), C07D 413/12 (2006.01), C07D 413/14 (2006.01), C07D 417/14 (2006.01), C07D 471/04 (2006.01)
Applicants: RAQUALIA PHARMA INC. [JP/JP]; 2, Aza 5-gochi, Taketoyo-cho, Chita-gun, Aichi 4702341 (JP) (For All Designated States Except US).
YAMAGISHI, Tatsuya [JP/JP]; (JP) (For US Only).
KAWAMURA, Kiyoshi [JP/JP]; (JP) (For US Only).
ARANO, Yoshimasa [JP/JP]; (JP) (For US Only).
MORITA, Mikio [JP/JP]; (JP) (For US Only)
Inventors: YAMAGISHI, Tatsuya; (JP).
KAWAMURA, Kiyoshi; (JP).
ARANO, Yoshimasa; (JP).
MORITA, Mikio; (JP)
Agent: IWATANI, Ryo; KEIHAN Dojima Bldg. 3F, 1-31, Dojima 2-chome, Kita-ku, Osaka-shi, Osaka 5300003 (JP)
Priority Data:
61/394,017 18.10.2010 US
61/418,002 30.11.2010 US
61/522,792 12.08.2011 US
Title (EN) ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS
(FR) DÉRIVÉS D'ARYLAMIDE EN TANT QU'AGENTS BLOQUANTS DE TTX-S
Abstract: front page image
(EN)The present invention relates to arylamide derivatives which have blocking activities of voltage gated sodium channels as the TTX-S channels, and which are useful in the treatment or prevention of disorders and diseases in which voltage gated sodium channels are involved. The invention also relates to pharmaceutical compositions comprising these compounds and the use of these compounds and compositions in the prevention or treatment of such diseases in which voltage gated sodium channels are involved.
(FR)La présente invention concerne des dérivés d'arylamide présentant des effets bloquants sur les canaux sodiques voltage-dépendants tels que les canaux TTX-S, et pouvant être employés dans le traitement prophylactique ou thérapeutique des troubles et maladies impliquant les canaux sodiques voltage-dépendants. La présente invention concerne également des compositions pharmaceutiques comprenant lesdits composés, ainsi que l'emploi desdits composés et compositions dans le traitement prophylactique ou thérapeutique de maladies impliquant les canaux sodiques voltage-dépendants.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)