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1. (WO2012052788) METHOD FOR PREPARING PHARMACEUTICALLY ACTIVE INGREDIENT AND INTERMEDIATES THEREOF
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2012/052788    International Application No.:    PCT/HU2011/000099
Publication Date: 26.04.2012 International Filing Date: 21.10.2011
IPC:
C07D 495/04 (2006.01), C07C 45/63 (2006.01)
Applicants: EGIS GYÓGYSZERGYÁR NYILVÁNOSAN MŰKÖDŐ RÉSZVÉNYTÁRSASÁG [HU/HU]; Keresztúri út 30-38 H-1106 Budapest (HU) (For All Designated States Except US).
NYULASI, Bálint [HU/HU]; (HU) (For US Only).
PORCS-MAKKAY, Márta [HU/HU]; (HU) (For US Only).
NÉMETH, Gábor [HU/HU]; (HU) (For US Only).
GREGOR, Tamás [HU/HU]; (HU) (For US Only).
BARKÓCZY, József [HU/HU]; (HU) (For US Only).
VOLK, Balázs [HU/HU]; (HU) (For US Only).
NAGY, Kálmán [HU/HU]; (HU) (For US Only).
RUZSICS, György [HU/HU]; (HU) (For US Only).
PAPP-FÜZFAI, Zsófia [HU/HU]; (HU) (For US Only).
MOLNÁR, Enikö [HU/HU]; (HU) (For US Only).
PANDUR, Angéla [HU/HU]; (HU) (For US Only).
KESZTHELYI, Adrienn [HU/HU]; (HU) (For US Only).
MEZEI, Tibor [HU/HU]; (HU) (For US Only).
FRIGYES, Dávid [HU/HU]; (HU) (For US Only)
Inventors: NYULASI, Bálint; (HU).
PORCS-MAKKAY, Márta; (HU).
NÉMETH, Gábor; (HU).
GREGOR, Tamás; (HU).
BARKÓCZY, József; (HU).
VOLK, Balázs; (HU).
NAGY, Kálmán; (HU).
RUZSICS, György; (HU).
PAPP-FÜZFAI, Zsófia; (HU).
MOLNÁR, Enikö; (HU).
PANDUR, Angéla; (HU).
KESZTHELYI, Adrienn; (HU).
MEZEI, Tibor; (HU).
FRIGYES, Dávid; (HU)
Agent: ADVOPATENT; Office of Patent and Trademark Attorneys P.O. Box 80 H-1255 Budapest (HU)
Priority Data:
P1000565 22.10.2010 HU
Title (EN) METHOD FOR PREPARING PHARMACEUTICALLY ACTIVE INGREDIENT AND INTERMEDIATES THEREOF
(FR) PROCÉDÉ DE PRÉPARATION D'UNE SUBSTANCE PHARMACEUTIQUEMENT ACTIVE ET DE SES INTERMÉDIAIRES
Abstract: front page image
(EN)The present invention is related to a safe and industrially applicable method for the preparation of 2-acetoxy-5-(2-fluoro-α-cyclopropyl- carbonyl-benzyl)-4,5,6,7-tetrahydro-4H-thieno[3,2-c]pyridine in a quality suitable for use as pharmaceutically active ingredient wherein the concentration of the impurities of the Formula.(XXIV) or (XXIVa) is reduced.
(FR)Cette invention concerne un procédé de préparation de 2-acétoxy- 5-(2-fluoro-α-cyclopropylcarbonylbenzyl)-4,5,6,7-tétrahydro-4H-thiéno-[3,2-c]pyridine, sans danger et industriellement applicable, à une qualité se prêtant à une utilisation à titre de substance pharmaceutiquement active, la concentration des impuretés dans ladite substance étant réduite. Formule (XXIV) ou (XXIVa).
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)