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Machine translation
1. (WO2012051036) QUINAZOLINONE-TYPE COMPOUNDS AS CRTH2 ANTAGONISTS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2012/051036    International Application No.:    PCT/US2011/055054
Publication Date: 19.04.2012 International Filing Date: 06.10.2011
IPC:
A01N 43/54 (2006.01), C07D 239/42 (2006.01), C07D 401/04 (2006.01)
Applicants: MERCK SHARP & DOHME CORP. [US/US]; 126 East Lincoln Avenue Rahway, New Jersey 07065-0907 (US) (For All Designated States Except US).
ASLANIAN, Robert, G. [US/US]; (US) (NZ, US only).
BOYCE, Christopher, W. [US/US]; (US) (NZ, US only).
MAZZOLA, Robert, D., Jr. [US/US]; (US) (NZ, US only).
MCKITTRICK, Brian, A. [US/US]; (US) (NZ, US only).
MCCORMICK, Kevin, D. [US/US]; (US) (NZ, US only).
PALANI, Anandan [US/US]; (US) (For US Only).
QIN, Jun [CN/US]; (US) (NZ, US only).
TANG, Haiqun [CN/US]; (US) (NZ, US only).
XIAO, Dong [CN/US]; (US) (NZ, US only).
YU, Younong [CN/US]; (US) (NZ, US only).
CALDWELL, John, P. [US/US]; (US) (NZ, US only).
KELLEY, Elizabeth Helen [US/US]; (US) (NZ, US only).
ZHANG, Hongjun [CN/US]; (US) (NZ, US only).
SILIPHAIVANH, Phieng [US/US]; (US) (NZ, US only).
MACCOSS, Rachel, N. [US/GB]; (GB) (NZ, US only).
METHOT, Joey, L. [US/US]; (US) (NZ, US only).
GAUUAN, Jolicia Polivina [US/US]; (US) (NZ, US only).
JIANG, Qin [US/US]; (US) (NZ, US only).
LEYHANE, Andrew, J. [US/US]; (US) (NZ, US only).
BIJU, Purakkattle Johny [US/US]; (US) (NZ, US only).
DONG, Li [CN/US]; (US) (NZ, US only).
HUANG, Xianhai [CN/US]; (US) (NZ, US only).
SHAO, Ning [CN/US]; (US) (NZ, US only).
ZHOU, Wei [US/US]; (US) (NZ, US only).
DHONDI, Pawan, K. [IN/US]; (US) (NZ, US only)
Inventors: ASLANIAN, Robert, G.; (US).
BOYCE, Christopher, W.; (US).
MAZZOLA, Robert, D., Jr.; (US).
MCKITTRICK, Brian, A.; (US).
MCCORMICK, Kevin, D.; (US).
PALANI, Anandan; (US).
QIN, Jun; (US).
TANG, Haiqun; (US).
XIAO, Dong; (US).
YU, Younong; (US).
CALDWELL, John, P.; (US).
KELLEY, Elizabeth Helen; (US).
ZHANG, Hongjun; (US).
SILIPHAIVANH, Phieng; (US).
MACCOSS, Rachel, N.; (GB).
METHOT, Joey, L.; (US).
GAUUAN, Jolicia Polivina; (US).
JIANG, Qin; (US).
LEYHANE, Andrew, J.; (US).
BIJU, Purakkattle Johny; (US).
DONG, Li; (US).
HUANG, Xianhai; (US).
SHAO, Ning; (US).
ZHOU, Wei; (US).
DHONDI, Pawan, K.; (US).
RAO, Ashwin, U.; (US)
Common
Representative:
MERCK SHARP & DOHME CORP.; 126 East Lincoln Avenue Rahway, New Jersey 07065-0907 (US)
Priority Data:
61/391,864 11.10.2010 US
Title (EN) QUINAZOLINONE-TYPE COMPOUNDS AS CRTH2 ANTAGONISTS
(FR) COMPOSÉS DE TYPE QUINAZOLINONE CONVENANT COMME ANTAGONISTES DE CRTH2
Abstract: front page image
(EN)This application provides for compounds of the formula Formula I or a pharmaceutically acceptable salt thereof, wherein the individual variables are defined herein, as well as processes to prepare these compounds, pharmaceutical compositions comprising the same and their use in treating disease state associated with the CRTH2 receptor.
(FR)La présente invention concerne des composés représentés par la formule (I), ou l'un de ses sels pharmaceutiquement admis, les différentes variables de cette formule étant telles que définies dans les spécifications. L'invention concerne également des procédés d'élaboration de ces composés, des compositions pharmaceutiques comprenant ces composés, et leur utilisation pour le traitement d'un état pathologique associé au récepteur du CRTH2.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)