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1. WO2012045124 - BACTERIA TOPOISOMERASE II INHIBITING 2-ETHYLCARBAMOYLAMINO-1, 3-BENZOTHIAZOL-5-YLS

Publication Number WO/2012/045124
Publication Date 12.04.2012
International Application No. PCT/AU2011/001284
International Filing Date 07.10.2011
IPC
C07D 417/14 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
417Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/196
14containing three or more hetero rings
A61K 31/429 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
41having five-membered rings with two or more ring hetero atoms, at least one of which is nitrogen, e.g. tetrazole
425Thiazoles
429condensed with heterocyclic ring systems
C07D 403/14 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
403Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/167
14containing three or more hetero rings
A61K 31/428 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
41having five-membered rings with two or more ring hetero atoms, at least one of which is nitrogen, e.g. tetrazole
425Thiazoles
428condensed with carbocyclic rings
A61P 31/04 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
31Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
04Antibacterial agents
C07D 413/14 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
413Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
14containing three or more hetero rings
CPC
A01N 47/36
AHUMAN NECESSITIES
01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES
47Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
08the carbon atom having one or more single bonds to nitrogen atoms
28Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
36containing the group >N—CO—N< directly attached to at least one heterocyclic ring; Thio analogues thereof
A61P 31/04
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
31Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
04Antibacterial agents
C07D 417/14
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
417Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
14containing three or more hetero rings
C07D 491/04
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
491Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
02in which the condensed system contains two hetero rings
04Ortho-condensed systems
C07D 513/04
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
513Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
02in which the condensed system contains two hetero rings
04Ortho-condensed systems
Applicants
  • BIOTA EUROPE LTD [GB]/[GB] (AllExceptUS)
  • PALMER, James T [US]/[AU] (UsOnly)
  • LUNNISS, Christopher James [GB]/[AU] (UsOnly)
  • OFFERMANN, Daniel A [AU]/[AU] (UsOnly)
  • AXFORD, Lorraine Claire [GB]/[AU] (UsOnly)
  • BLAIR, Michael [AU]/[AU] (UsOnly)
  • MITCHELL, Dale Robert [GB]/[GB] (UsOnly)
  • PALMER, Nicholas John [GB]/[GB] (UsOnly)
  • STEELE, Christopher [GB]/[GB] (UsOnly)
  • ATHERALL, John [GB]/[GB] (UsOnly)
  • WATSON, David [GB]/[GB] (UsOnly)
  • HAYDON, David John [GB]/[GB] (UsOnly)
  • CZAPLEWSKI, Lloyd George [GB]/[GB] (UsOnly)
  • DAVIES, David [GB]/[GB] (UsOnly)
  • COLLINS, Ian [GB]/[GB] (UsOnly)
  • TYNDALL, Edward Malcolm (UsOnly)
  • ANDRAU, Laura (UsOnly)
  • PITT, Gary Robert William (UsOnly)
Inventors
  • PALMER, James T
  • LUNNISS, Christopher James
  • OFFERMANN, Daniel A
  • AXFORD, Lorraine Claire
  • BLAIR, Michael
  • MITCHELL, Dale Robert
  • PALMER, Nicholas John
  • STEELE, Christopher
  • ATHERALL, John
  • WATSON, David
  • HAYDON, David John
  • CZAPLEWSKI, Lloyd George
  • DAVIES, David
  • COLLINS, Ian
  • TYNDALL, Edward Malcolm
  • ANDRAU, Laura
  • PITT, Gary Robert William
Agents
  • FB RICE
Priority Data
61/391,16308.10.2010US
Publication Language English (en)
Filing Language English (EN)
Designated States
Title
(EN) BACTERIA TOPOISOMERASE II INHIBITING 2-ETHYLCARBAMOYLAMINO-1, 3-BENZOTHIAZOL-5-YLS
(FR) 2-ÉTHYLCARBAMOYLAMINO-1,3-BENZOTHIAZOL-5-YLES INHIBITEURS DE TOPOISOMÉRASE II BACTÉRIENNE
Abstract
(EN) The present invention provides a compound of the following formula and salts thereof: Also provided is the use of these compounds as antibacterials, compositions comprising them and processes for their manufacture.
(FR) La présente invention concerne un composé de formule suivante et ses sels : La présente invention concerne également l'emploi desdits composés comme antibactériens, les compositions les incluant et leurs procédés de fabrication.
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