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1. (WO2012045124) BACTERIA TOPOISOMERASE II INHIBITING 2-ETHYLCARBAMOYLAMINO-1, 3-BENZOTHIAZOL-5-YLS
Latest bibliographic data on file with the International Bureau   

Pub. No.: WO/2012/045124 International Application No.: PCT/AU2011/001284
Publication Date: 12.04.2012 International Filing Date: 07.10.2011
IPC:
C07D 417/14 (2006.01) ,A61K 31/429 (2006.01) ,C07D 403/14 (2006.01) ,A61K 31/428 (2006.01) ,A61P 31/04 (2006.01) ,C07D 413/14 (2006.01) ,C07D 471/04 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
417
Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/196
14
containing three or more hetero rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
41
having five-membered rings with two or more ring hetero atoms, at least one of which is nitrogen, e.g. tetrazole
425
Thiazoles
429
condensed with heterocyclic ring systems
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
403
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/167
14
containing three or more hetero rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
41
having five-membered rings with two or more ring hetero atoms, at least one of which is nitrogen, e.g. tetrazole
425
Thiazoles
428
condensed with carbocyclic rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
31
Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
04
Antibacterial agents
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
413
Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
14
containing three or more hetero rings
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
471
Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/-C07D463/251
02
in which the condensed system contains two hetero rings
04
Ortho-condensed systems
Applicants:
PALMER, James T [US/AU]; AU (UsOnly)
LUNNISS, Christopher James [GB/AU]; AU (UsOnly)
OFFERMANN, Daniel A [AU/AU]; AU (UsOnly)
AXFORD, Lorraine Claire [GB/AU]; AU (UsOnly)
BLAIR, Michael [AU/AU]; AU (UsOnly)
MITCHELL, Dale Robert [GB/GB]; GB (UsOnly)
PALMER, Nicholas John [GB/GB]; GB (UsOnly)
STEELE, Christopher [GB/GB]; GB (UsOnly)
ATHERALL, John [GB/GB]; GB (UsOnly)
WATSON, David [GB/GB]; GB (UsOnly)
HAYDON, David John [GB/GB]; GB (UsOnly)
CZAPLEWSKI, Lloyd George [GB/GB]; GB (UsOnly)
DAVIES, David [GB/GB]; GB (UsOnly)
COLLINS, Ian [GB/GB]; GB (UsOnly)
TYNDALL, Edward Malcolm; AU (UsOnly)
ANDRAU, Laura; AU (UsOnly)
PITT, Gary Robert William; AU (UsOnly)
BIOTA EUROPE LTD [GB/GB]; Begbroke Business & Science Park Sandy Lane Yarnton Oxfordshire OX5 1PF, GB (AllExceptUS)
Inventors:
PALMER, James T; AU
LUNNISS, Christopher James; AU
OFFERMANN, Daniel A; AU
AXFORD, Lorraine Claire; AU
BLAIR, Michael; AU
MITCHELL, Dale Robert; GB
PALMER, Nicholas John; GB
STEELE, Christopher; GB
ATHERALL, John; GB
WATSON, David; GB
HAYDON, David John; GB
CZAPLEWSKI, Lloyd George; GB
DAVIES, David; GB
COLLINS, Ian; GB
TYNDALL, Edward Malcolm; AU
ANDRAU, Laura; AU
PITT, Gary Robert William; AU
Agent:
FB RICE; Level 23 200 Queen Street Melbourne, Victoria 3000, AU
Priority Data:
61/391,16308.10.2010US
Title (EN) BACTERIA TOPOISOMERASE II INHIBITING 2-ETHYLCARBAMOYLAMINO-1, 3-BENZOTHIAZOL-5-YLS
(FR) 2-ÉTHYLCARBAMOYLAMINO-1,3-BENZOTHIAZOL-5-YLES INHIBITEURS DE TOPOISOMÉRASE II BACTÉRIENNE
Abstract:
(EN) The present invention provides a compound of the following formula and salts thereof: Also provided is the use of these compounds as antibacterials, compositions comprising them and processes for their manufacture.
(FR) La présente invention concerne un composé de formule suivante et ses sels : La présente invention concerne également l'emploi desdits composés comme antibactériens, les compositions les incluant et leurs procédés de fabrication.
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Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)