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1. (WO2012042915) SULFAMOYL BENZOIC ACID HETEROBICYCLIC DERIVATIVES AS TRPM8 ANTAGONISTS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2012/042915    International Application No.:    PCT/JP2011/005588
Publication Date: 05.04.2012 International Filing Date: 03.10.2011
IPC:
C07D 401/12 (2006.01), A61K 31/443 (2006.01), A61K 31/4439 (2006.01), A61K 31/444 (2006.01), A61K 31/4709 (2006.01), A61P 13/00 (2006.01), A61P 25/00 (2006.01), A61P 29/00 (2006.01), A61P 43/00 (2006.01), C07D 209/08 (2006.01), C07D 215/12 (2006.01), C07D 231/56 (2006.01), C07D 249/18 (2006.01), C07D 307/79 (2006.01), C07D 405/04 (2006.01), C07D 405/12 (2006.01), C07D 405/14 (2006.01), C07D 471/04 (2006.01)
Applicants: RAQUALIA PHARMA INC. [JP/JP]; 2, Aza 5-gochi, Taketoyo-cho, Chita-gun, Aichi 4702341 (JP) (For All Designated States Except US).
KAWAMURA, Kiyoshi [JP/JP]; (JP) (For US Only).
SHISHIDO, Yuji [JP/JP]; (JP) (For US Only).
OHMI, Masashi [JP/JP]; (JP) (For US Only)
Inventors: KAWAMURA, Kiyoshi; (JP).
SHISHIDO, Yuji; (JP).
OHMI, Masashi; (JP)
Agent: IWATANI, Ryo; KEIHAN Dojima Bldg. 3F, 1-31, Dojima 2-chome, Kita-ku, Osaka-shi, Osaka 5300003 (JP)
Priority Data:
61/388,696 01.10.2010 US
Title (EN) SULFAMOYL BENZOIC ACID HETEROBICYCLIC DERIVATIVES AS TRPM8 ANTAGONISTS
(FR) DÉRIVÉS HÉTÉROBICYCLIQUES D'ACIDE SULFAMOYLBENZOÏQUE EN TANT QU'ANTAGONISTES DE TRPM8
Abstract: front page image
(EN)The present invention relates to sulfamoyl benzoic acid heterobicyclic derivatives of the formula (I) or a pharmaceutically acceptable salt thereof or a prodrug thereof, processes for their preparation, pharmaceutical compositions containing them and their use in the treatment of various disorders which are mediated via the TRPM8 receptor.
(FR)La présente invention concerne des dérivés hétérobicycliques d'acide sulfamoylbenzoïque de formule (I) ou un de leurs sels pharmaceutiquement acceptables ou promédicaments, leurs procédés de préparation, des compositions pharmaceutiques les contenant et leur utilisation dans le traitement de divers troubles médiés par le récepteur TRPM8.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)