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Machine translation
1. (WO2012042482) PROCESS FOR THE SYNTHESIS OF FUNICONE ANALOGUES
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2012/042482    International Application No.:    PCT/IB2011/054262
Publication Date: 05.04.2012 International Filing Date: 28.09.2011
IPC:
C07D 309/38 (2006.01), C07C 49/503 (2006.01), A61K 31/351 (2006.01), A61P 31/00 (2006.01), A61P 35/00 (2006.01)
Applicants: CONSIGLIO NAZIONALE DELLE RICERCHE [IT/IT]; Piazzale Aldo Moro, 7 I-00185 Roma (IT) (For All Designated States Except US).
CONSIGLIO PER LA RICERCA E LA SPERIMENTAZIONE IN AGRICOLTURA [IT/IT]; Via Nazionale, 82 I-00184 Roma (IT) (For All Designated States Except US).
MANZO, Emiliano [IT/IT]; (IT) (For US Only).
CIAVATTA, Maria, Letizia [IT/IT]; (IT) (For US Only).
NICOLETTI, Rosario [IT/IT]; (IT) (For US Only)
Inventors: MANZO, Emiliano; (IT).
CIAVATTA, Maria, Letizia; (IT).
NICOLETTI, Rosario; (IT)
Agent: FINETTI, Claudia; c/o Barzano' & Zanardo Milano S.p.A. Via Borgonuovo, 10 I-20121 Milano (IT)
Priority Data:
MI2010A 001770 28.09.2010 IT
Title (EN) PROCESS FOR THE SYNTHESIS OF FUNICONE ANALOGUES
(FR) PROCÉDÉ POUR LA SYNTHÈSE D'ANALOGUES DE FUNICONE
Abstract: front page image
(EN)The present invention relates to the synthesis of analogous compounds of funicone, some of which are not found in nature, which comprises the preparation of compounds having general formula (III) and (IV) and the subsequent coupling reaction of said compounds in dimethylformamide by means of carbon monoxide in the presence of palladium allyl chloride dimer, to obtain compounds having formula (V) (scheme 2).
(FR)L'invention concerne la synthèse de composés analogues de funicone, dont certains ne se trouvent pas dans la nature, qui fait appel à la préparation de composés de formules générales (III) et (IV) et à la réaction de couplage subséquente desdits composés en diméthylformamide au moyen de monoxyde de carbone en présence d'un dimère de chlorure d'allyle palladium, pour obtenir des composés de formule (V) (schéma 2).
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: Italian (IT)