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1. (WO2011162222) NOVEL CRYSTALLINE FORMS OF 4,4'-[4-FLUORO-7-({4-[4-(3-FLUORO-2-METHYLPHENYL)BUTOXY]PHENYL}ETHYNYL)-2-METHYL-1H-INDOLE-1,3-DIYL]DIBUTANOIC ACID, 4,4'-[2-METHYL-7-({4-[4-(PENTAFLUOROPHENYL)BUTOXY]PHENYL}ETHYNYL)-1H-INDOLE-1,3-DIYL]DIBUTANOIC ACID, AND 4,4'-[4-FLUORO-2-METHYL-7-({4-[4-(2,3,4,6-TETRAFLUOROPHENYL)BUTOXY]PHENYL}ETHYNYL)-1H-INDOLE-1,3-DIYL]DIBUTANOIC ACID
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2011/162222    International Application No.:    PCT/JP2011/064088
Publication Date: 29.12.2011 International Filing Date: 20.06.2011
IPC:
C07D 209/18 (2006.01), A61K 31/405 (2006.01), A61P 11/06 (2006.01), A61P 37/08 (2006.01), A61P 43/00 (2006.01)
Applicants: ONO PHARMACEUTICAL CO., LTD. [JP/JP]; 1-5, Doshomachi 2-chome, Chuo-ku, Osaka-shi, Osaka 5418526 (JP) (For All Designated States Except US).
TAKEUCHI, Jun [JP/JP]; (JP) (For US Only).
ITADANI, Satoshi [JP/JP]; (JP) (For US Only).
UEDA, Junya [JP/JP]; (JP) (For US Only).
ONO, Shizuka [JP/JP]; (JP) (For US Only).
NEKADO, Takahiro [JP/JP]; (JP) (For US Only).
FUJITA, Manabu [JP/JP]; (JP) (For US Only)
Inventors: TAKEUCHI, Jun; (JP).
ITADANI, Satoshi; (JP).
UEDA, Junya; (JP).
ONO, Shizuka; (JP).
NEKADO, Takahiro; (JP).
FUJITA, Manabu; (JP)
Agent: AOKI, Atsushi; SEIWA PATENT & LAW, Toranomon 37 Mori Bldg., 5-1, Toranomon 3-chome, Minato-ku, Tokyo 1058423 (JP)
Priority Data:
2010-140344 21.06.2010 JP
Title (EN) NOVEL CRYSTALLINE FORMS OF 4,4'-[4-FLUORO-7-({4-[4-(3-FLUORO-2-METHYLPHENYL)BUTOXY]PHENYL}ETHYNYL)-2-METHYL-1H-INDOLE-1,3-DIYL]DIBUTANOIC ACID, 4,4'-[2-METHYL-7-({4-[4-(PENTAFLUOROPHENYL)BUTOXY]PHENYL}ETHYNYL)-1H-INDOLE-1,3-DIYL]DIBUTANOIC ACID, AND 4,4'-[4-FLUORO-2-METHYL-7-({4-[4-(2,3,4,6-TETRAFLUOROPHENYL)BUTOXY]PHENYL}ETHYNYL)-1H-INDOLE-1,3-DIYL]DIBUTANOIC ACID
(FR) NOUVELLE FORME CRISTALLINE D'ACIDE DIBUTANOÏQUE 4, 4'-[4-FLUORO-7-({4-[4-(3-FLUORO-2-MÉTHYLPHÉNYL) BUTOXY] PHÉNYL} ÉTHYNYLE)-2-MÉTHYLE-1H-INDOLE-1,3-DIYLE], D'ACIDE DIBUTANOÏQUE 4, 4'-[2-MÉTHYLE-7-({4-[4-(PENTAFLUOROPHÉNYL) BUTOXY] PHÉNYL} ÉTHYNYLE)-1H-INDOLE-1,3-DIYLE], ET D'ACIDE DIBUTANOÏQUE 4, 4'-[4-FLUORO-2-MÉTHYLE-7-({4-[4-(2, 3, 4, 6-TÉTRAFLUOROPHÉNYL) BUTOXY] PHÉNYL} ÉTHYNYLE)-1H-INDOLE-1,3-DIYLE]
(JA) 4,4'-[4-フルオロ-7-({4-[4-(3-フルオロ-2-メチルフェニル)ブトキシ]フェニル}エチニル)-2-メチル-1H-インドール-1,3-ジイル]ジブタン酸、4,4'-[2-メチル-7-({4-[4-(ペンタフルオロフェニル)ブトキシ]フェニル}エチニル)-1H-インドール-1,3-ジイル]ジブタン酸および4,4'-[4-フルオロ-2-メチル-7-({4-[4-(2,3,4,6-テトラフルオロフェニル)ブトキシ]フェニル}エチニル)-1H-インドール-1,3-ジイル]ジブタン酸の新規結晶形
Abstract: front page image
(EN)Provided are a C-form crystal of compound (I), a B-form crystal of compound (II), and a C-form crystal of compound (III), as set forth in the Description.
(FR)La présente invention concerne un cristal de forme C d'un composé (I), un cristal de forme B d'un composé (II) et un cristal de forme C d'un composé (III).
(JA) 本明細書で示される化合物IのC型結晶、化合物IIのB型結晶および化合物IIIのC型結晶の提供。
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: Japanese (JA)
Filing Language: Japanese (JA)