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1. (WO2011145669) AMIDE DERIVATIVE
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2011/145669    International Application No.:    PCT/JP2011/061473
Publication Date: 24.11.2011 International Filing Date: 19.05.2011
IPC:
C07C 233/11 (2006.01), A61K 31/341 (2006.01), A61K 31/343 (2006.01), A61K 31/351 (2006.01), A61K 31/38 (2006.01), A61K 31/397 (2006.01), A61K 31/40 (2006.01), A61K 31/402 (2006.01), A61K 31/4152 (2006.01), A61K 31/4164 (2006.01), A61K 31/4166 (2006.01), A61K 31/4192 (2006.01), A61K 31/421 (2006.01), A61K 31/4245 (2006.01), A61K 31/426 (2006.01), A61K 31/428 (2006.01), A61K 31/44 (2006.01), A61K 31/4402 (2006.01), A61K 31/4406 (2006.01), A61K 31/4409 (2006.01), A61K 31/47 (2006.01), A61K 31/4965 (2006.01), A61K 31/50 (2006.01), A61K 31/505 (2006.01), A61P 25/00 (2006.01), A61P 25/08 (2006.01), C07C 233/65 (2006.01), C07C 311/13 (2006.01), C07C 311/16 (2006.01), C07D 205/04 (2006.01), C07D 207/04 (2006.01), C07D 207/27 (2006.01), C07D 207/28 (2006.01), C07D 207/333 (2006.01), C07D 207/408 (2006.01), C07D 213/30 (2006.01), C07D 213/34 (2006.01), C07D 213/36 (2006.01), C07D 213/50 (2006.01), C07D 213/56 (2006.01), C07D 213/61 (2006.01), C07D 213/65 (2006.01), C07D 213/82 (2006.01), C07D 215/12 (2006.01), C07D 231/12 (2006.01), C07D 231/34 (2006.01), C07D 233/34 (2006.01), C07D 233/64 (2006.01), C07D 233/70 (2006.01), C07D 233/74 (2006.01), C07D 233/76 (2006.01), C07D 237/08 (2006.01), C07D 239/26 (2006.01), C07D 241/12 (2006.01), C07D 241/24 (2006.01), C07D 249/04 (2006.01), C07D 263/20 (2006.01), C07D 263/22 (2006.01), C07D 263/32 (2006.01), C07D 263/44 (2006.01), C07D 265/32 (2006.01), C07D 271/06 (2006.01), C07D 271/10 (2006.01), C07D 277/20 (2006.01), C07D 277/24 (2006.01), C07D 277/26 (2006.01), C07D 277/28 (2006.01), C07D 277/30 (2006.01), C07D 277/56 (2006.01), C07D 277/66 (2006.01), C07D 307/38 (2006.01), C07D 307/42 (2006.01), C07D 307/52 (2006.01), C07D 307/68 (2006.01), C07D 309/06 (2006.01), C07D 333/16 (2006.01), C07D 333/18 (2006.01), C07D 333/38 (2006.01), C07D 333/56 (2006.01)
Applicants: Dainippon Sumitomo Pharma Co., Ltd. [JP/JP]; 6-8, Dosho-machi 2-chome, Chuo-ku, Osaka-shi, Osaka 5418524 (JP) (For All Designated States Except US).
IWAMA, Seiji [JP/JP]; (JP) (For US Only).
TANAKA, Tomoyuki [JP/JP]; (JP) (For US Only).
GOTOH, Nana [JP/JP]; (JP) (For US Only)
Inventors: IWAMA, Seiji; (JP).
TANAKA, Tomoyuki; (JP).
GOTOH, Nana; (JP)
Agent: TANAKA, Mitsuo; AOYAMA & PARTNERS IMP Building 3-7, Shiromi 1-chome, Chuo-ku Osaka-shi, Osaka 5400001 (JP)
Priority Data:
2010-115010 19.05.2010 JP
Title (EN) AMIDE DERIVATIVE
(FR) DÉRIVÉ D'AMIDE
(JA) アミド誘導体
Abstract: front page image
(EN)Disclosed are the compound represented by formula (I) which is useful as a therapeutic or prophylactic agent for various partial and/or generalized epileptic seizures, or a salt thereof. [In the formula, ring A and ring B independently represent aryl rings, L represents a bond, a C1-6 alkylene, etc., Alk represents a bond, a C1-6 alkylene, etc., X represents -CONR7R8, -SO2NR7R8, etc., R1, R2, and R3 are the same or different and represent a hydrogen atom, a halogen, etc., R4 and R5 independently represent a hydrogen atom, a halogen, etc., and R7 and R8, etc., independently represent a hydrogen atom, a C1-6 alkyl, etc.]
(FR)La présente invention concerne le composé représenté par la formule (I) qui est utile en tant qu'agent thérapeutique ou prophylactique pour différentes crises épileptiques partielles et/ou généralisées, ou un sel de celui-ci. [Dans la formule, le cycle A et le cycle B représentent indépendamment des cycles aryle, L représente une liaison, un alkylène en C1-6, etc., Alk représente une liaison, un alkylène en C1-6, etc., X représente -CONR7R8, -SO2NR7R8, etc., R1, R2, et R3 sont identiques ou différents et représentent un atome d'hydrogène, un halogène, etc., R4 et R5 représentent indépendamment un atome d'hydrogène, un halogène, etc., et R7 et R8, etc., représentent indépendamment un atome d'hydrogène, un alkyle en C1-6, etc.]
(JA) 本発明は、部分発作及び/又は全般発作の種々てんかん発作に対する治療薬若しくは予防薬として有用な式(I)の化合物又はその塩[式中、A環及びB環は、それぞれ独立して、アリール環等を表し、Lは、結合、C1-6アルキレン等を表し、Alkは、結合、C1-6アルキレン等を表し、Xは、-CONR、-SONR等を表し、R、R及びRは、同一又は異なって、水素原子、ハロゲン等を表し、R及びRは、それぞれ独立して、水素原子、ハロゲン等を表し、R、R等は、それぞれ独立して、水素原子、C1-6アルキル等を表す]を提供する。
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: Japanese (JA)
Filing Language: Japanese (JA)