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1. (WO2011143106) BI - FUNCTIONAL PYRAZOLOPYRIDINE COMPOUNDS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2011/143106    International Application No.:    PCT/US2011/035741
Publication Date: 17.11.2011 International Filing Date: 09.05.2011
IPC:
C07D 471/04 (2006.01), A61K 31/437 (2006.01), A61P 29/00 (2006.01), A61P 37/08 (2006.01)
Applicants: GILEAD SCIENCES, INC. [US/US]; 333 Lakeside Drive Foster City, CA 94404 (US) (For All Designated States Except US).
BAKER, William, R. [US/US]; (US) (For US Only).
CAI, Shaopei [US/US]; (US) (For US Only).
KAPLAN, Joshua, Aaron [US/US]; (US) (For US Only).
KIM, Musong [US/US]; (US) (For US Only).
PHILLIPS, Gary [US/US]; (US) (For US Only).
PURVIS, II., Lafe, J. [US/US]; (US) (For US Only).
STASIAK, Marcin [US/US]; (US) (For US Only).
STEVENS, Kirk, L. [US/US]; (US) (For US Only).
VAN VELDHUIZEN, Josh [US/US]; (US) (For US Only)
Inventors: BAKER, William, R.; (US).
CAI, Shaopei; (US).
KAPLAN, Joshua, Aaron; (US).
KIM, Musong; (US).
PHILLIPS, Gary; (US).
PURVIS, II., Lafe, J.; (US).
STASIAK, Marcin; (US).
STEVENS, Kirk, L.; (US).
VAN VELDHUIZEN, Josh; (US)
Agent: ECK, Steven, R.; Gilead Sciences, Inc. 333 Lakeside Drive Foster City, CA 94404 (US)
Priority Data:
61/333,031 10.05.2010 US
61/406,933 26.10.2010 US
61/477,264 20.04.2011 US
Title (EN) BI - FUNCTIONAL PYRAZOLOPYRIDINE COMPOUNDS
(FR) COMPOSÉS PYRAZOLOPYRIDINIQUES BIFONCTIONNELS
Abstract: front page image
(EN)invention provides compounds of the formula: wherein R1 and R2 together with the phenyl to which they are bound may form a bicyclic, fused heterocyclic ring and all other variables are as defined herein, their use in pulmonary inflammation or bronchoconstriction therapy and compositions comprising and processes for preparing the same are provided.
(FR)La présente invention concerne, des composés représentés par la formule (I), dans laquelle R1 et R2 forment ensemble, avec le phényle auquel ils sont liés, un noyau hétérocyclique fusionné bicyclique, et toutes les autres variables sont telles que définies dans la présente demande. L'invention concerne également l'utilisation de ces composés pour le traitement de l'inflammation pulmonaire ou de la bronchoconstriction, et des compositions comprenant ces composés, et leurs procédés de préparation.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)