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1. (WO2011137220) SMALL MOLECULE NEUROPEPTIDE S ANTAGONISTS FOR THE TREATMENT OF ADDICTIVE DISORDERS, MOOD, ANXIETY AND SLEEP DISORDERS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2011/137220    International Application No.:    PCT/US2011/034276
Publication Date: 03.11.2011 International Filing Date: 28.04.2011
IPC:
C07D 209/08 (2006.01), C07D 209/42 (2006.01), C07F 9/547 (2006.01), C07F 9/553 (2006.01)
Applicants: THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES [US/US]; Office of Technology Transfer National Institutes of Health 6011 Executive Boulevard, Suite 325 MSC 7660 Bethesda, Maryland 20892-7660 (US) (For All Designated States Except US).
MARUGAN, Juan J. [US/US]; (US) (For US Only).
PATNAIK, Samarjit [IN/US]; (US) (For US Only).
HEILIG, Markus A. [SE/US]; (US) (For US Only).
SOUTHALL, Noel T. [US/US]; (US) (For US Only).
ZHENG, Wei [US/US]; (US) (For US Only)
Inventors: MARUGAN, Juan J.; (US).
PATNAIK, Samarjit; (US).
HEILIG, Markus A.; (US).
SOUTHALL, Noel T.; (US).
ZHENG, Wei; (US)
Agent: CONTRERA, Joseph G.; Leydig, Voit & Mayer Two Prudential Plaza, Suite 4900 180 North Stetson Avenue Chicago, Illinois 60601-6731 (US)
Priority Data:
61/328,900 28.04.2010 US
Title (EN) SMALL MOLECULE NEUROPEPTIDE S ANTAGONISTS FOR THE TREATMENT OF ADDICTIVE DISORDERS, MOOD, ANXIETY AND SLEEP DISORDERS
(FR) ANTAGONISTES À PETITE MOLÉCULE DU NEUROPEPTIDE S DESTINÉS AU TRAITEMENT D'UNE TOXICOMANIE OU DE TROUBLES DE L'HUMEUR, DE L'ANXIÉTÉ ET DU SOMMEIL
Abstract: front page image
(EN)Disclosed are compounds of General Formula I: wherein R1, R2, R3, X and Y are described herein, as well as pharmaceutically acceptable salts, solvates, and stereoisomers thereof. Pharmaceutical compositions comprising such compounds, as well as methods of use, and treatment for neuropsychiatric disorders including pain, sleep, mood, anxiety, eating and addictive disorders, are also provided.
(FR)La présente invention concerne des composés de formule générale I : dans laquelle R1, R2, R3, X et Y sont décrits dans ce document, ainsi que leurs sels pharmaceutiquement acceptables, solvates et stéréo-isomères. L'invention concerne également des compositions pharmaceutiques contenant ces composés ainsi que des méthodes d'utilisation et de traitement de troubles neuropsychiatriques y compris la douleur, des troubles du sommeil, de l'humeur, de l'anxiété, de l'alimentation et de toxicomanie.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)