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1. WO2011133888 - CERTAIN AMINO-PYRIMIDINES, COMPOSITIONS THEREOF, AND METHODS FOR THEIR USE

Publication Number WO/2011/133888
Publication Date 27.10.2011
International Application No. PCT/US2011/033614
International Filing Date 22.04.2011
IPC
A61K 31/4965 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
495having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
4965Non-condensed pyrazines
CPC
A61K 9/0014
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
9Medicinal preparations characterised by special physical form
0012Galenical forms characterised by the site of application
0014Skin, i.e. galenical aspects of topical compositions
A61K 9/0019
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
9Medicinal preparations characterised by special physical form
0012Galenical forms characterised by the site of application
0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
A61K 9/0034
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
9Medicinal preparations characterised by special physical form
0012Galenical forms characterised by the site of application
0034Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
A61K 9/0043
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
9Medicinal preparations characterised by special physical form
0012Galenical forms characterised by the site of application
0043Nose
A61K 9/0048
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
9Medicinal preparations characterised by special physical form
0012Galenical forms characterised by the site of application
0048Eye, e.g. artificial tears
A61K 9/0053
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
9Medicinal preparations characterised by special physical form
0012Galenical forms characterised by the site of application
0053Mouth and digestive tract, i.e. intraoral and peroral administration
Applicants
  • CYTOKINETICS, INC. [US]/[US] (AllExceptUS)
  • YANG, Zhe [US]/[US] (UsOnly)
  • MUCI, Alex R. [US]/[US] (UsOnly)
  • WARRINGTON, Jeffrey [CA]/[US] (UsOnly)
  • BERGNES, Gustave [US]/[US] (UsOnly)
  • MORGAN, Bradley P. [US]/[US] (UsOnly)
  • CHUANG, Chihyuan [US]/[US] (UsOnly)
  • ROMERO, Antonio [US]/[US] (UsOnly)
  • COLLIBEE, Scott [US]/[US] (UsOnly)
  • QIAN, Xiangping [US]/[US] (UsOnly)
  • LU, Pu-Ping [US]/[US] (UsOnly)
Inventors
  • YANG, Zhe
  • MUCI, Alex R.
  • WARRINGTON, Jeffrey
  • BERGNES, Gustave
  • MORGAN, Bradley P.
  • CHUANG, Chihyuan
  • ROMERO, Antonio
  • COLLIBEE, Scott
  • QIAN, Xiangping
  • LU, Pu-Ping
Agents
  • STEVENS, Lauren
Priority Data
61/327,59723.04.2010US
61/412,29910.11.2010US
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) CERTAIN AMINO-PYRIMIDINES, COMPOSITIONS THEREOF, AND METHODS FOR THEIR USE
(FR) CERTAINES AMINO-PYRIDAZINES, COMPOSITIONS CONTENANT CES DERNIÈRES ET LEURS PROCÉDÉS D'UTILISATION
Abstract
(EN)
Provided are compounds of Formula (I) or a pharmaceutically acceptable salt thereof, wherein R1, R2, R3, R4, R5, R6, R7, R8, R9, X and m are as defined herein. Also provided is a pharmaceutically acceptable composition comprising a compound of Formula I, or a pharmaceutically acceptable salt thereof. Also provided are methods of using a compound of Formula I, or a pharmaceutically acceptable salt thereof.
(FR)
L'invention concerne des composés de Formule I : (I) ou un sel pharmaceutiquement acceptable de ceux-ci. Dans la formule, R1, R2, R3, R4, R5, R6, R7, R8, R9, X et m sont tels que définis dans la description. L'invention concerne également une composition pharmaceutiquement acceptable comprenant un composé de Formule I, ou un sel pharmaceutiquement acceptable de celui-ci. L'invention concerne aussi des procédés d'utilisation d'un composé de Formule I ou d'un sel pharmaceutiquement acceptable de celui-ci.
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