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1. WO2011060391 - SELECTIVE HETEROCYCLIC SPHINGOSINE 1 PHOSPHATE RECEPTOR MODULATORS

Publication Number WO/2011/060391
Publication Date 19.05.2011
International Application No. PCT/US2010/056759
International Filing Date 15.11.2010
IPC
A01N 43/78 2006.1
AHUMAN NECESSITIES
01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
72having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms
74five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
781,3-Thiazoles; Hydrogenated 1,3-thiazoles
A61K 31/425 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
41having five-membered rings with two or more ring hetero atoms, at least one of which is nitrogen, e.g. tetrazole
425Thiazoles
CPC
A61K 2300/00
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
2300Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
A61K 31/433
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
41having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
433Thidiazoles
A61K 45/06
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
45Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
A61P 1/04
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
1Drugs for disorders of the alimentary tract or the digestive system
04for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
A61P 11/00
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
11Drugs for disorders of the respiratory system
A61P 25/00
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
25Drugs for disorders of the nervous system
Applicants
  • RECEPTOS, INC. [US]/[US] (AllExceptUS)
  • BOEHM, Marcus, F. [US]/[US] (UsOnly)
  • MARTINBOROUGH, Esther [US]/[US] (UsOnly)
  • BRAHMACHARY, Enugurthi [IN]/[US] (UsOnly)
  • MOORJANI, Manisha [CA]/[US] (UsOnly)
  • TAMIYA, Junko (UsOnly)
  • HUANG, Liming (UsOnly)
  • YEAGER, Adam, Richard (UsOnly)
Inventors
  • BOEHM, Marcus, F.
  • MARTINBOROUGH, Esther
  • BRAHMACHARY, Enugurthi
  • MOORJANI, Manisha
  • TAMIYA, Junko
  • HUANG, Liming
  • YEAGER, Adam, Richard
Agents
  • BLAYLOCK, Richard, L.
Priority Data
61/261,29513.11.2009US
61/262,47418.11.2009US
Publication Language English (en)
Filing Language English (EN)
Designated States
Title
(EN) SELECTIVE HETEROCYCLIC SPHINGOSINE 1 PHOSPHATE RECEPTOR MODULATORS
(FR) MODULATEURS DE RÉCEPTEUR DE SPHINGOSINE-1-PHOSPHATE HÉTÉROCYCLIQUES SÉLECTIFS
Abstract
(EN) Compounds that selectively modulate the sphingosine 1 phosphate receptor are provided including compounds which modulate subtype 1 of the SlP receptor. Methods of chiral synthesis of such compounds is provided. Uses, methods of treatment or prevention and methods of preparing inventive compositions including inventive compounds are provided in connection with the treatment or prevention of diseases, malconditions, and disorders for which modulation of the sphingosine 1 phosphate receptor is medically indicated.
(FR) La présente invention concerne des composés qui modulent sélectivement le récepteur de sphingosine-1-phosphate, y compris des composés qui modulent le sous-type 1 du récepteur S1P. La présente invention concerne des procédés de synthèse chirale de tels composés. La présente invention concerne des utilisations, des méthodes de traitement ou de prévention et des procédés de préparation de compositions de l'invention comprenant des composés de l'invention dans le contexte du traitement ou de la prévention de maladies, affections, et troubles pour lesquels la modulation du récepteur de sphingosine-1-phosphate est médicalement indiquée.
Related patent documents
MXMX/a/2012/005559This application is not viewable in PATENTSCOPE because the national phase entry has not been published yet or the national entry is issued from a country that does not share data with WIPO or there is a formatting issue or an unavailability of the application.
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