WIPO logo
Mobile | Deutsch | Español | Français | 日本語 | 한국어 | Português | Русский | 中文 | العربية |
PATENTSCOPE

Search International and National Patent Collections
World Intellectual Property Organization
Search
 
Browse
 
Translate
 
Options
 
News
 
Login
 
Help
 
Machine translation
1. (WO2011019612) BORON-CONTAINING SMALL MOLECULES AS ANTIPROTOZOAL AGENTS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2011/019612    International Application No.:    PCT/US2010/044727
Publication Date: 17.02.2011 International Filing Date: 06.08.2010
IPC:
A61K 31/69 (2006.01), C07F 5/02 (2006.01), A61P 33/02 (2006.01)
Applicants: ANACOR PHARMACEUTICALS, INC. [US/US]; 1020 East Meadow Circle Palo Alto, CA 94303 (US) (For All Designated States Except US).
ORR, Matthew [US/US]; (US) (For US Only).
JENKS, Matthew [US/US]; (US) (For US Only)
Inventors: ORR, Matthew; (US).
JENKS, Matthew; (US)
Agent: ESKER, Todd; Morgan, Lewis & Bockius, LLP One Marker, Spear Street Tower San Francisco, CA 94105 (US)
Priority Data:
61/308,717 26.02.2010 US
61/234,222 14.08.2009 US
Title (EN) BORON-CONTAINING SMALL MOLECULES AS ANTIPROTOZOAL AGENTS
(FR) PETITES MOLÉCULES CONTENANT DU BORE EN TANT QU'AGENTS ANTIPROTOZOAIRES
Abstract: front page image
(EN)This invention provides, among other things, novel compounds useful for treating protozoal infections, pharmaceutical compositions containing such compounds, as well as combinations of these compounds with at least one additional therapeutically effective agent. The compounds are of formula (I), wherein Z is S or O; and X is selected from the group consisting of substituted phenyl, substituted or unsubstituted heteroaryl, and unsubstituted cycloalkyl, or a salt thereof.
(FR)L'invention concerne, entre autres, de nouveaux composés utiles pour traiter les infections protozoaires, des compositions pharmaceutiques contenant lesdits composés, ainsi que des combinaisons de ces composés avec au moins un agent supplémentaire thérapeutiquement efficace. Les composés sont de formule (I), où Z représente S ou O; et X est choisi dans le groupe constitué par le phényle substitué, l'hétéroaryle substitué ou non substitué et le cycloalkyle non substitué, ou un sel de ceux-ci.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)