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1. (WO2011015037) ANTIVIRAL COMPOUNDS AND METHODS OF MAKING AND USING THEREOF
Latest bibliographic data on file with the International Bureau   

Pub. No.: WO/2011/015037 International Application No.: PCT/CN2010/001187
Publication Date: 10.02.2011 International Filing Date: 05.08.2010
Chapter 2 Demand Filed: 19.04.2011
IPC:
C07D 413/12 (2006.01) ,C07D 295/00 (2006.01) ,A61K 31/497 (2006.01) ,A61K 31/44 (2006.01) ,A61K 31/42 (2006.01) ,A61K 31/00 (2006.01) ,A61P 31/16 (2006.01) ,A61P 31/12 (2006.01)
Applicants: KAO, Yitsun, Richard[CN/CN]; CN (UsOnly)
YANG, Dan[CN/CN]; CN (UsOnly)
YEUN, Kwokyung[CN/CN]; CN (UsOnly)
VERSITECH LIMITED[CN/CN]; Finance Office The University of Hong Kong Pokfulam Road Hong Kong, CN (AllExceptUS)
Inventors: KAO, Yitsun, Richard; CN
YANG, Dan; CN
YEUN, Kwokyung; CN
Agent: CHINA PATENT AGENT (H. K.) LTD.; 22/F, Great Eagle Centre 23 Harbour Road, Wanchai Hong Kong, CN
Priority Data:
61/231, 43105.08.2009US
Title (EN) ANTIVIRAL COMPOUNDS AND METHODS OF MAKING AND USING THEREOF
(FR) COMPOSÉS ANTIVIRAUX ET LEURS PROCÉDÉS DE FABRICATION ET D'UTILISATION
Abstract:
(EN) Compounds which exhibit antiviral activity, particularly against influenza virus,and methods of making and using there of are described herein. In one embodiment, the compounds are heterocyclic amides containing piperazine and isozazole rings and optionally substituted with one or more substituents. The compounds can be formulated with one or more pharmaceutically acceptable excipients to form compositions suitable for enteralor parenteral administration. The compounds are preferably used to treat or prevent Influenza Ainfections, such as H1N1, H2N2, H3N2, H5N1, H7N7, H1N2, H9N2, H7N2, H7N3, and H10N7.
(FR) L'invention porte sur des composés qui présentent une activité antivirale, en particulier contre le virus de la grippe, et sur leurs procédés de fabrication et d'utilisation. Dans un mode de réalisation, les composés sont des amides hétérocycliques contenant des noyaux pipérazine et isoxazole et faculatativement substitués par un ou plusieurs substituants. Les composés peuvent être formulés avec un ou plusieurs excipients de qualité pharmaceutique pour former des compositions appropriées pour l'administration entérale ou parentérale. Les composés sont de préférence utilisés pour traiter ou prévenir des infections de type grippe A, telles que H1N1, H2N2, H3N2, H5N1, H7N7, H1N2, H9N2, H7N2, H7N3 et H10N7.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)