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1. WO2011006569 - HETEROCYCLIC COMPOUNDS AS AUTOTAXIN INHIBITORS

Publication Number WO/2011/006569
Publication Date 20.01.2011
International Application No. PCT/EP2010/003661
International Filing Date 17.06.2010
IPC
C07D 487/04 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
487Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/-C07D477/183
02in which the condensed system contains two hetero rings
04Ortho-condensed systems
C07D 487/14 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
487Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/-C07D477/183
12in which the condensed system contains three hetero rings
14Ortho-condensed systems
A61K 31/5513 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
55having seven-membered rings, e.g. azelastine, pentylenetetrazole
551having two nitrogens as ring hetero atoms, e.g. clozapine, dilazep
55131,4-Benzodiazepines, e.g. diazepam
A61P 35/00 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
35Antineoplastic agents
CPC
A61P 35/00
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
35Antineoplastic agents
A61P 35/02
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
35Antineoplastic agents
02specific for leukemia
A61P 43/00
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
43Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
C07D 487/04
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
487Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by C07D451/00 - C07D477/00
02in which the condensed system contains two hetero rings
04Ortho-condensed systems
Applicants
  • MERCK PATENT GMBH [DE]/[DE] (AllExceptUS)
  • SCHULTZ, Melanie [DE]/[DE] (UsOnly)
  • SCHIEMANN, Kai [DE]/[DE] (UsOnly)
  • STAEHLE, Wolfgang [DE]/[DE] (UsOnly)
Inventors
  • SCHULTZ, Melanie
  • SCHIEMANN, Kai
  • STAEHLE, Wolfgang
Common Representative
  • MERCK PATENT GMBH [DE]/[DE]
Priority Data
10 2009 033 392.416.07.2009DE
Publication Language German (DE)
Filing Language German (DE)
Designated States
Title
(DE) HETEROCYCLISCHE VERBINDUNGEN ALS AUTOTAXIN-INHIBITOREN
(EN) HETEROCYCLIC COMPOUNDS AS AUTOTAXIN INHIBITORS
(FR) COMPOSÉS HÉTÉROCYCLIQUES EN TANT QU'INHIBITEURS D'AUTOTAXINE
Abstract
(DE)
Verbindungen der Formel (I) worin R, R1, R2, X, X1, Y, Y1, Q, E, n1 und n2 die in Anspruch 1 angegebenen Bedeutungen haben, sind Autotaxin-Inhibitoren und können zur Behandlung von Tumoren eingesetzt werden.
(EN)
Compounds of the formula (I), where R1, R2, X, X1, Y, Y1, Q, E, n1 and n2 have the meanings indicated in claim 1, are autotaxin inhibitors and can be used for the treatment of tumors.
(FR)
L'invention concerne des composés de formule (I), dans laquelle R, R1, R2, X, X1, Y, Y1, Q, E, n1 et n2 ont les significations données dans la revendication 1. Ces composés sont des inhibiteurs d'autotaxine et peuvent être utilisés pour le traitement de tumeurs.
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