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1. (WO2010148396) PERINDOPRIL TOSYLATE
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2010/148396    International Application No.:    PCT/US2010/039350
Publication Date: 23.12.2010 International Filing Date: 21.06.2010
IPC:
C07D 209/42 (2006.01), A61K 31/404 (2006.01), A61P 9/12 (2006.01)
Applicants: TEVA PHARMACEUTICAL INDUSTRIES LTD. [IL/IL]; 5 Basel Street P.O. Box 3190 Petah Tiqva 49131 (IL) (AE, AG, AL, AM, AO, AT, AU, AZ, BA, BE, BF, BG, BH, BJ, BR, BW, BY, BZ, CA, CF, CG, CH, CI, CL, CM, CN, CO, CR, CU, CY, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, FR, GA, GB, GD, GE, GH, GM, GN, GQ, GR, GT, GW, HN, HR, HU, ID, IE, IL, IN, IS, IT, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LV, LY, MA, MC, MD, ME, MG, MK, ML, MN, MR, MT, MW, MX, MY, MZ, NA, NE, NG, NI, NL, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SI, SK, SL, SM, SN, ST, SV, SY, SZ, TD, TG, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, UZ, VC, VN, ZA, ZM, ZW only).
TEVA PHARMACEUTICALS USA, INC. [US/US]; 1090 Horsham Road P.O. Box 1090 North Wales, PA 19454-1090 (US) (BB only).
COSTI, Sonia [IL/IL]; (IL) (For US Only).
KHAN, Mubeen [IN/IN]; (IN) (For US Only).
GHARPURE, Milind [IN/IN]; (IN) (For US Only).
PANDEY, Anand, Kumar [IN/IN]; (IN) (For US Only).
YADAV, Roop Singh [IN/IN]; (IN) (For US Only).
PATIL, Pramod Vittal [IN/IN]; (IN) (For US Only).
LAD, Sachin [IN/IN]; (IN) (For US Only).
PATLE, Girish [IN/IN]; (IN) (For US Only)
Inventors: COSTI, Sonia; (IL).
KHAN, Mubeen; (IN).
GHARPURE, Milind; (IN).
PANDEY, Anand, Kumar; (IN).
YADAV, Roop Singh; (IN).
PATIL, Pramod Vittal; (IN).
LAD, Sachin; (IN).
PATLE, Girish; (IN)
Agent: BIRDE, Patrick, J.; Kenyon & Kenyon LLP One Broadway New York, NY 1004-1050 (US)
Priority Data:
0910692.3 20.06.2009 GB
Title (EN) PERINDOPRIL TOSYLATE
(FR) TOSYLATE DE PÉRINDOPRIL
Abstract: front page image
(EN)The present invention relates to a novel salt of perindopril, namely the paratoluene sulfonic acid salt. The present invention also relates to an amorphous form of the perindopril paratoluene sulfonic acid salt. The invention further relates to processes for the preparation of the novel salt and the amorphous form thereof. The invention also relates to pharmaceutical compositions comprising the perindopril tosylate for the treatment of hypertension and heart failure.
(FR)La présente invention concerne un nouveau sel de périndopril, à savoir le sel d'acide paratoluène sulfonique. L'invention porte en outre sur une forme amorphe du sel d'acide paratoluène sulfonique de périndopril. L'invention concerne également des méthodes de préparation du nouveau sel et de la forme amorphe de celui-ci. L'invention porte en outre sur des compositions pharmaceutiques comprenant le tosylate de périndopril, utilisées dans le traitement de l'hypertension et de l'insuffisance cardiaque.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)