WIPO logo
Mobile | Deutsch | Español | Français | 日本語 | 한국어 | Português | Русский | 中文 | العربية |
PATENTSCOPE

Search International and National Patent Collections
World Intellectual Property Organization
Search
 
Browse
 
Translate
 
Options
 
News
 
Login
 
Help
 
Machine translation
1. (WO2010147302) NOVEL INTERMEDIATES OF VORICONAZOLE AND PREPARATION METHOD OF VORICONAZOLE USING THE SAME
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2010/147302    International Application No.:    PCT/KR2010/002715
Publication Date: 23.12.2010 International Filing Date: 29.04.2010
IPC:
C07D 401/06 (2006.01), A61K 31/4196 (2006.01), A61K 31/506 (2006.01), A61K 47/40 (2006.01)
Applicants: BORYUNG PHARMACEUTICAL CO., LTD. [KR/KR]; 66-21, Wonnam-dong, Jongno-gu, Seoul 110-750 (KR) (For All Designated States Except US).
CHOI, Ok Kyoung [KR/KR]; (KR) (For US Only).
PARK, Yong [KR/KR]; (KR) (For US Only).
LEE, Joon Kwang [KR/KR]; (KR) (For US Only).
KIM, Ji Han [KR/KR]; (KR) (For US Only).
TAN, Hyun Kwang [KR/KR]; (KR) (For US Only)
Inventors: CHOI, Ok Kyoung; (KR).
PARK, Yong; (KR).
LEE, Joon Kwang; (KR).
KIM, Ji Han; (KR).
TAN, Hyun Kwang; (KR)
Agent: AHN, So-Young; Dr. Ahn International Patent Law Office 10th Fl., Shinseung Bldg., 1676-1, Seocho-dong, Seocho-gu, Seoul 137-881 (KR)
Priority Data:
10-2009-0053670 17.06.2009 KR
Title (EN) NOVEL INTERMEDIATES OF VORICONAZOLE AND PREPARATION METHOD OF VORICONAZOLE USING THE SAME
(FR) NOUVEAUX INTERMÉDIAIRES DE VORICONAZOLE ET PROCÉDÉ DE PRÉPARATION DE VORICONAZOLE LES UTILISANT
(KO) 보리코나졸의 신규 중간체 및 이를 이용한 보리코나졸의 제조방법
Abstract: front page image
(EN)The present invention provides compounds of Formulas 2 and 4 as novel intermediates of Voriconazole, and a preparation method of Voriconazole using the same. The novel intermediates of the present invention are environmentally friendly because pungent and unpleasant odors particular to thiols are eliminated, and allow Voriconazole to be prepared at high purities and high yields.
(FR)La présente invention porte sur des composés des Formules 2 et 4 en tant que nouveaux intermédiaires de Voriconazole, et sur un procédé de préparation de Voriconazole les utilisant. Les nouveaux intermédiaires de la présente invention sont écologiques parce que les odeurs piquantes et déplaisantes en particulier dues aux thiols sont éliminées, et permettent au Voriconazole d'être préparé à des puretés élevées et dans des rendements élevés.
(KO)본 발명은 보나코나졸의 신규한 중간체인 화학식 2 화합물, 화학식 4 화합물 및 이를 이용한 보리코나졸의 제조방법을 제공한다. 본 발명의 신규한 중간체는 티 올류 특유의 자극적이고 불쾌한 냄새가 배제된 것으로 친환경적임과 동시에 고순도 고수율로 보리코나졸을 제조하게 한다.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: Korean (KO)
Filing Language: Korean (KO)