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1. (WO2010143803) NEW NICOTINAMIDE DERIVATIVES WITH ANTI-ANDROGEN EFFECTS, PROCESSES OF PREPARING, AND ANTIANDROGENS COMPRISING THE SAME
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2010/143803    International Application No.:    PCT/KR2010/000960
Publication Date: 16.12.2010 International Filing Date: 17.02.2010
IPC:
C07D 213/81 (2006.01), C07D 403/10 (2006.01), C07D 487/04 (2006.01), C07D 403/12 (2006.01), A61K 31/4375 (2006.01), A61P 5/28 (2006.01)
Applicants: INDUSTRY FOUNDATION OF CHONNAM NATIONAL UNIVERSITY [KR/KR]; 300, Yongbong-dong, Buk-gu Gwangju 500-843 (KR) (For All Designated States Except US).
LEE, Keesook [KR/KR]; (KR) (For US Only).
SONG, Chin-Hee [KR/KR]; (KR) (For US Only).
CHO, Won-Jea [KR/KR]; (KR) (For US Only)
Inventors: LEE, Keesook; (KR).
SONG, Chin-Hee; (KR).
CHO, Won-Jea; (KR)
Agent: KWON, Oh-Sig; 4F, Jooeunleaderstel, 921, Dunsan-dong, Seo-gu Daejeon 302-120 (KR)
Priority Data:
10-2009-0050320 08.06.2009 KR
10-2009-0069557 29.07.2009 KR
Title (EN) NEW NICOTINAMIDE DERIVATIVES WITH ANTI-ANDROGEN EFFECTS, PROCESSES OF PREPARING, AND ANTIANDROGENS COMPRISING THE SAME
(FR) NOUVEAUX DÉRIVÉS DE NICOTINAMIDE AYANT DES EFFETS ANTI-ANDROGÉNIQUES, PROCÉDÉS DE PRÉPARATION, ET ANTI-ANDROGÈNES LES COMPRENANT
Abstract: front page image
(EN)Provided are novel nicotinamide derivatives and pharmaceutically acceptable salts thereof with anti-androgen effects, preparing processes of the same and antiandrogens containing the same as active ingredients. More particularly, the said nicotinamide derivatives have anti-androgen activity, so that they can be effectively used as a preventive or therapeutic agent for androgen-related diseases such as prostatic disease, androgenic alopecia and acne.
(FR)La présente invention concerne de nouveaux dérivés du nicotinamide ainsi que leurs sels pharmaceutiquement acceptables avec des effets anti-androgènes, leurs procédés de préparation et des anti-androgènes les contenant comme principes actifs. Plus particulièrement, lesdits dérivés du nicotinamide présentent une activité anti-androgénique, de telle sorte qu'ils peuvent être utilisés de façon efficace comme agents préventifs ou thérapeutiques dans les pathologies liées aux androgènes telles que la maladie de la prostate, l'alopécie androgénique et l'acné.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)