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Machine translation
1. (WO2010143735) METHOD FOR PRODUCING 4-SUBSTITUTED BENZOTHIOAMIDE DERIVATIVE
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2010/143735    International Application No.:    PCT/JP2010/060003
Publication Date: 16.12.2010 International Filing Date: 08.06.2010
IPC:
C07C 327/48 (2006.01)
Applicants: TEIJIN PHARMA LIMITED [JP/JP]; 2-1, Kasumigaseki 3-chome, Chiyoda-ku, Tokyo 1000013 (JP) (For All Designated States Except US).
SUGIURA, Satoshi [JP/JP]; (JP) (For US Only)
Inventors: SUGIURA, Satoshi; (JP)
Agent: MIHARA, Hideko; c/o Teijin Intellectual Property Center Limited, 2-1, Kasumigaseki 3-chome, Chiyoda-ku, Tokyo 1000013 (JP)
Priority Data:
2009-138049 09.06.2009 JP
Title (EN) METHOD FOR PRODUCING 4-SUBSTITUTED BENZOTHIOAMIDE DERIVATIVE
(FR) PROCÉDÉ DE FABRICATION D'UN DÉRIVÉ DE BENZOTHIOAMIDE 4-SUBSTITUÉ
(JA) 4-置換ベンゾチオアミド誘導体の製造法
Abstract: front page image
(EN)Disclosed is a method appropriate for safely, economically and easily producing at a high yield a 4-substituted benzothioamide derivative which is useful as an intermediate in the production of a 2-(3-cyanophenyl)thiazole derivative usable as a remedy for gout. Specifically disclosed is a method for producing a 4-substituted benzothioamide derivative represented by formula (A).
(FR)L'invention porte sur un procédé apte à produire d'une manière sûre, économique et aisée, avec un rendement élevé, un dérivé de benzothioamide 4-substitué, qui est utile en tant qu'intermédiaire de la production d'un dérivé du 2-(3-cyanophényl)thiazole, pouvant être utilisé en tant que remède pour la goutte. De façon spécifique, l'invention porte sur un procédé de production d'un dérivé de benzothioamide 4-substitué de formule (A).
(JA)本発明の課題は、痛風治療薬として使用される2-(3-シアノフェニル)チアゾール誘導体の、製造中間体として有用な4-置換ベンゾチオアミド誘導体を、安全、安価、容易且つ高収率に製造するのに適した方法を提供することである。本発明は、下記式で表される4-置換ベンゾチオアミド誘導体の製造方法に関する。
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: Japanese (JA)
Filing Language: Japanese (JA)