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1. WO2010093419 - NOVEL AMINO AZAHETEROCYCLIC CARBOXAMIDES

Publication Number WO/2010/093419
Publication Date 19.08.2010
International Application No. PCT/US2010/000313
International Filing Date 04.02.2010
IPC
C07D 239/94 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
239Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
70condensed with carbocyclic rings or ring systems
72Quinazolines; Hydrogenated quinazolines
86with hetero atoms directly attached in position 4
94Nitrogen atoms
C07D 401/04 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
401Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
02containing two hetero rings
04directly linked by a ring-member-to-ring- member bond
C07D 401/12 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
401Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
02containing two hetero rings
12linked by a chain containing hetero atoms as chain links
C07D 403/12 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
403Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/167
02containing two hetero rings
12linked by a chain containing hetero atoms as chain links
C07D 405/12 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
405Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
02containing two hetero rings
12linked by a chain containing hetero atoms as chain links
C07D 409/04 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
409Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
02containing two hetero rings
04directly linked by a ring-member-to-ring- member bond
CPC
A61K 31/47
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
435having six-membered rings with one nitrogen as the only ring hetero atom
47Quinolines; Isoquinolines
A61P 1/18
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
1Drugs for disorders of the alimentary tract or the digestive system
18for pancreatic disorders, e.g. pancreatic enzymes
A61P 13/12
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
13Drugs for disorders of the urinary system
12of the kidneys
A61P 17/00
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
17Drugs for dermatological disorders
A61P 17/06
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
17Drugs for dermatological disorders
06Antipsoriatics
A61P 25/04
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
25Drugs for disorders of the nervous system
04Centrally acting analgesics, e.g. opioids
Applicants
  • MERCK PATENT GMBH [DE]/[DE] (AllExceptUS)
  • SUTTON, Amanda E. [US]/[US] (UsOnly)
  • RICHARDSON, Thomas E. [US]/[US] (UsOnly)
  • HUCK, Bayard R. [US]/[US] (UsOnly)
  • KARRA, Srinivasa R. [IN]/[US] (UsOnly)
  • CHEN, Xiaoling [CA]/[US] (UsOnly)
  • XIAO, Yufang [CA]/[US] (UsOnly)
  • GOUTOPOULOS, Andreas [GR]/[US] (UsOnly)
  • LAN, Ruoxi [CA]/[US] (UsOnly)
  • PERREY, David [GB]/[US] (UsOnly)
  • VANDEVEER, Harold, George [US]/[US] (UsOnly)
  • LIU-BUJALSKI, Lesley [CA]/[US] (UsOnly)
  • STIEBER, Frank [DE]/[DE] (UsOnly)
  • HODOUS, Brian L. [US]/[US] (UsOnly)
  • QIU, Hui [CN]/[US] (UsOnly)
  • JONES, Reinaldo C. [US]/[US] (UsOnly)
  • HEASLEY, Brian [US]/[US] (UsOnly)
Inventors
  • SUTTON, Amanda E.
  • RICHARDSON, Thomas E.
  • HUCK, Bayard R.
  • KARRA, Srinivasa R.
  • CHEN, Xiaoling
  • XIAO, Yufang
  • GOUTOPOULOS, Andreas
  • LAN, Ruoxi
  • PERREY, David
  • VANDEVEER, Harold, George
  • LIU-BUJALSKI, Lesley
  • STIEBER, Frank
  • HODOUS, Brian L.
  • QIU, Hui
  • JONES, Reinaldo C.
  • HEASLEY, Brian
Agents
  • SEEMANN, PH.D., Joachim
Priority Data
61/207,35411.02.2009US
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) NOVEL AMINO AZAHETEROCYCLIC CARBOXAMIDES
(FR) NOUVEAUX CARBOXAMIDES AMINO-AZAHÉTÉROCYCLIQUES
Abstract
(EN)
The invention provides novel substituted amino azaheterocyclic carboxamide compounds according to Formula (I), their manufacture and use for the treatment of hyperproliferative diseases, such as cancer.
(FR)
L'invention concerne de nouveaux composés de carboxamide amino-azahétérocyclique substitué selon la formule (I), leur fabrication et utilisation pour le traitement de maladies hyperprolifératives, telles que le cancer.
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