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1. (WO2010086349) ANTI-INFLAMMATORY MACROLIDE
Latest bibliographic data on file with the International Bureau   

Pub. No.: WO/2010/086349 International Application No.: PCT/EP2010/050967
Publication Date: 05.08.2010 International Filing Date: 28.01.2010
Chapter 2 Demand Filed: 30.11.2010
IPC:
C07H 17/08 (2006.01) ,A61K 31/7048 (2006.01) ,A61P 29/00 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
H
SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
17
Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
04
Heterocyclic radicals containing only oxygen as ring hetero atoms
08
Hetero rings containing eight or more ring members, e.g. erythromycins
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
70
Carbohydrates; Sugars; Derivatives thereof
7042
Compounds having saccharide radicals and heterocyclic rings
7048
having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
29
Non-central analgesic, antipyretic or antiinflammatory agents, e.g antirheumatic agents; Non-steroidal antiinflammatory drugs (NSAIDs)
Applicants:
DAY, Caroline, Jane [GB/GB]; GB (UsOnly)
DOUILLET, Julien, Bruno [FR/GB]; GB (UsOnly)
FILIC, Darko [HR/HR]; GB (UsOnly)
KINDON, Leanda, Jane [GB/GB]; GB (UsOnly)
KRAGOL, Goran [HR/HR]; GB (UsOnly)
MARUSIC-ISTUK, Zorica [HR/HR]; GB (UsOnly)
GLAXO GROUP LIMITED [GB/GB]; Glaxo Wellcome House Berkeley Avenue Greenford Middlesex UB6 0NN, GB (AllExceptUS)
Inventors:
DAY, Caroline, Jane; GB
DOUILLET, Julien, Bruno; GB
FILIC, Darko; GB
KINDON, Leanda, Jane; GB
KRAGOL, Goran; GB
MARUSIC-ISTUK, Zorica; GB
Agent:
CRAWLEY, Karen; GlaxoSmithKline Corporate Intellectual Property CN925.1 980 Great West Road Brentford Middlesex TW8 9GS, GB
Priority Data:
61/148,60930.01.2009US
Title (EN) ANTI-INFLAMMATORY MACROLIDE
(FR) MACROLIDE ANTI-INFLAMMATOIRE
Abstract:
(EN) The compound 3'-N-demethyl-4"-O-(2-diethylaminoethanoyl)-6-O-methyl-9a-aza-9a- homoerythromycin A, having the Formula (I): or a salt thereof, compositions comprising the compound, its use in the treatment of neutrophil dominated inflammatory diseases, and methods for its preparation.
(FR) La présente invention porte sur le composé 3'-N-déméthyl-4''-O-(2-diéthylaminoéthanoyl)-6-O-méthyl-9a-aza-9a-homoérythromycine A, répondant à la formule (I) ou un sel de celui-ci, sur des compositions comprenant le composé, sur ses utilisations pour le traitement de maladies inflammatoires dominées par les neutrophiles et sur ses procédés de préparation.
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Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)