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1. (WO2010079120) BENZIMIDAZOLE AND PYRAZOLOPYRIDINE DERIVATIVES FOR TREATING AND/OR PREVENTING CARDIOVASCULAR DISEASES
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2010/079120 International Application No.: PCT/EP2010/000011
Publication Date: 15.07.2010 International Filing Date: 05.01.2010
IPC:
C07D 403/04 (2006.01) ,C07D 403/14 (2006.01) ,C07D 471/04 (2006.01) ,A61K 31/506 (2006.01) ,A61P 9/00 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
403
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/167
02
containing two hetero rings
04
directly linked by a ring-member-to-ring- member bond
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
403
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/167
14
containing three or more hetero rings
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
471
Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/-C07D463/251
02
in which the condensed system contains two hetero rings
04
Ortho-condensed systems
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
495
having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
505
Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
506
not condensed and containing further heterocyclic rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
9
Drugs for disorders of the cardiovascular system
Applicants:
BAYER PHARMA AKTIENGESELLSCHAFT [DE/DE]; Müllerstr. 178 13353 Berlin, DE (AllExceptUS)
STRAUB, Alexander [DE/DE]; DE (UsOnly)
SÜßMEIER, Frank [DE/DE]; DE (UsOnly)
WUNDER, Frank [DE/DE]; DE (UsOnly)
STASCH, Johannes-Peter [DE/DE]; DE (UsOnly)
LI, Volkhart, Min-Jian [DE/DE]; DE (UsOnly)
MITTENDORF, Joachim [DE/DE]; DE (UsOnly)
Inventors:
STRAUB, Alexander; DE
SÜßMEIER, Frank; DE
WUNDER, Frank; DE
STASCH, Johannes-Peter; DE
LI, Volkhart, Min-Jian; DE
MITTENDORF, Joachim; DE
Common
Representative:
BAYER PHARMA AKTIENGESELLSCHAFT [DE/DE]; Law and Patents, Patents and Licensing 51368 Leverkusen, DE
Priority Data:
10 2009 004 245.809.01.2009DE
Title (DE) BENZIMIDAZOL-UND PYRAZOLOPYRIDIN-DERIVATE ZUR BEHANDLUNG UND/ODER PRÄVENTION VON HERZ-KREISLAUF-ERKRANKUNGEN
(EN) BENZIMIDAZOLE AND PYRAZOLOPYRIDINE DERIVATIVES FOR TREATING AND/OR PREVENTING CARDIOVASCULAR DISEASES
(FR) DÉRIVÉS DE BENZIMIDAZOLE ET PYRAZOLOPYRIDINE POUR LE TRAITEMENT ET/OU LA PRÉVENTION DE MALADIES CARDIOVASCULAIRES
Abstract:
(DE) Die vorliegende Anmeldung betrifft neue Benzimidazol-und Pyrazolopyridin derivate, Verfahren zu ihrer Herstellung, ihre Verwendung allein oder in Kombinationen zur Behandlung und/oder Prävention von Krankheiten sowie ihre Verwendung zur Herstellung von Arzneimitteln zur Behandlung und/oder Prävention von Krankheiten, insbesondere zur Behandlung und/oder Prävention von Herz-Kreislauf-Erkrankungen.
(EN) The present invention relates to novel benzimidazole and pyrazolopyridine derivatives, to methods for the production thereof, to the use thereof alone or in combination to treat and/or prevent illnesses, and to the use thereof to produce drugs for treating and/or preventing illnesses, in particular for treating and/or preventing cardiovascular diseases.
(FR) La présente invention porte sur de nouveaux dérivés de benzimidazole et pyrazolopyridine, sur un procédé permettant de les fabriquer, sur leur utilisation individuellement ou dans des combinaisons pour le traitement et/ou la prévention de maladie ainsi que sur leur utilisation pour la fabrication de médicaments pour le traitement et/ou la prévention de maladies, en particulier pour le traitement et/ou la prévention de maladies cardiovasculaires.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: German (DE)
Filing Language: German (DE)
Also published as:
EP2385942US20120029002CA2749048US20130303559