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1. (WO2010078830) BENZIMIDAZOLE-4-CARBOXAMIDE DERIVATIVES, THEIR PREPARATION METHODS, PHARMACEUTICAL COMPOSITIONS AND THEIR USES
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2010/078830 International Application No.: PCT/CN2010/000024
Publication Date: 15.07.2010 International Filing Date: 06.01.2010
IPC:
C07D 401/12 (2006.01) ,C07D 405/12 (2006.01) ,C07D 403/12 (2006.01) ,C07D 417/12 (2006.01) ,A61K 31/4184 (2006.01) ,A61K 31/4439 (2006.01) ,A61P 31/12 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
401
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
02
containing two hetero rings
12
linked by a chain containing hetero atoms as chain links
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
405
Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
02
containing two hetero rings
12
linked by a chain containing hetero atoms as chain links
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
403
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/167
02
containing two hetero rings
12
linked by a chain containing hetero atoms as chain links
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
417
Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/196
02
containing two hetero rings
12
linked by a chain containing hetero atoms as chain links
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
41
having five-membered rings with two or more ring hetero atoms, at least one of which is nitrogen, e.g. tetrazole
4164
1,3-Diazoles
4184
condensed with carbocyclic rings, e.g. benzimidazoles
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
435
having six-membered rings with one nitrogen as the only ring hetero atom
44
Non-condensed pyridines; Hydrogenated derivatives thereof
4427
containing further heterocyclic ring systems
4439
containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
31
Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
12
Antivirals
Applicants:
上海交通大学 SHANGHAI JIAO TONG UNIVERSITY [CN/CN]; 中国上海市华山路1954号, Shanghai 200240 No. 1954, Hua Shan Road Shanghai 200240, CN (AllExceptUS)
罗先金 LUO, Xianjin [CN/CN]; CN (UsOnly)
薛飞 XUE, Fei [CN/CN]; CN (UsOnly)
张钟闾 ZHANG, Zhonglv [CN/CN]; CN (UsOnly)
修乃云 XIU, Naiyun [CN/CN]; CN (UsOnly)
Inventors:
罗先金 LUO, Xianjin; CN
薛飞 XUE, Fei; CN
张钟闾 ZHANG, Zhonglv; CN
修乃云 XIU, Naiyun; CN
Agent:
北京乾诚五洲知识产权代理有限责任公司 FAITHFULAW INTERNATIONAL IP LAW OFFICE; 中国北京市西城区北三环中路甲29号3号楼A-1101室, Beijing 100029 Suite 1101, Block A, Building No. 3 A29, Beisanhuanzhonglu, Xicheng District Beijing 100029, CN
Priority Data:
200910045056.808.01.2009CN
201010000050.105.01.2010CN
Title (EN) BENZIMIDAZOLE-4-CARBOXAMIDE DERIVATIVES, THEIR PREPARATION METHODS, PHARMACEUTICAL COMPOSITIONS AND THEIR USES
(FR) DÉRIVÉS DE BENZIMIDAZOLE-4-CARBOXAMIDE, LEURS PROCÉDÉS D'ÉLABORATION, COMPOSITIONS PHARMACEUTIQUES ET LEURS UTILISATIONS
(ZH) 苯并咪唑-4-酰胺型衍生物及其制备方法、药物组合物及其用途
Abstract:
(EN) The benzimidazole-4-carboxamide derivatives of formula (Ⅰ) in which X and Y are defined as the specification, their preparation methods, pharmaceutical compositions and their uses are disclosed. The derivatives of the present invention have antiviral activity.
(FR) La présente invention concerne des dérivés de benzimidazole-4-carboxamide représentés par la formule (I) dans laquelle X et Y sont tels que définis dans les spécifications. L'invention concerne également leurs procédés d'élaboration, des compositions pharmaceutiques, et leurs utilisations. Les dérivés de la présente invention sont dotés d'activité antivirale.
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Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: Chinese (ZH)
Filing Language: Chinese (ZH)
Also published as:
EP2386553JP2012514607US20110269766RU2011133009CA2749174KR1020110124751
EP2963033AU2010204407IN6012/DELNP/2011