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1. (WO2010077758) COMPOUNDS USEFUL FOR INHIBITING CHK1
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2010/077758 International Application No.: PCT/US2009/067437
Publication Date: 08.07.2010 International Filing Date: 10.12.2009
IPC:
C07D 403/12 (2006.01) ,A61K 31/497 (2006.01) ,A61P 35/00 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
403
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/167
02
containing two hetero rings
12
linked by a chain containing hetero atoms as chain links
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
495
having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
4965
Non-condensed pyrazines
497
containing further heterocyclic rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
35
Antineoplastic agents
Applicants:
ELI LILLY AND COMPANY [US/US]; Lilly Corporate Center Indianapolis, Indiana 46285, US (AllExceptUS)
FAROUZ, Francine, S. [FR/US]; US (UsOnly)
HOLCOMB, Ryan, Coatsworth [US/US]; US (UsOnly)
KASAR, Ramesh [US/US]; US (UsOnly)
MYERS, Steven, Scott [US/US]; US (UsOnly)
Inventors:
FAROUZ, Francine, S.; US
HOLCOMB, Ryan, Coatsworth; US
KASAR, Ramesh; US
MYERS, Steven, Scott; US
Agent:
HOSTETTLER, Danica; ELI LILLY AND COMPANY Patent Division P. O. Box 6288 Indianapolis, Indiana 46206-6288, US
Priority Data:
61/138,17617.12.2008US
Title (EN) COMPOUNDS USEFUL FOR INHIBITING CHK1
(FR) COMPOSÉS UTILES POUR INHIBER CHK1
Abstract:
(EN) The present invention provides an aminopyrazole compound, or a pharmaceutically acceptable salt thereof or a solvate of the salt, that inhibits Chk1 and is useful in the treatment of cancer.
(FR) La présente invention porte sur un composé aminopyrazole ou sur un sel de qualité pharmaceutique de celui-ci ou sur un solvate du sel, qui inhibe Chk1 et qui s'utilise dans le traitement du cancer.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)
Also published as:
RSP-2013/0153UAa201107564PA20098850801AR074471DOP2011000185IL213160
SG172222EP2379532MA32901JP2012512249ES2401558CN102245597
CA2746423EA201170834MX2011006603KR1020110084539TN2011000298NZ593440
AU2009333433DK2379532VN27547BNRE/2015/0006ID051.4894MYPI 2011002767
TH128480IN4123/CHENP/2011