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1. (WO2010076813) THIENOPYRIDINES AS PHARMACOLOGICALLY ACTIVE AGENTS
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2010/076813 International Application No.: PCT/IN2010/000005
Publication Date: 08.07.2010 International Filing Date: 05.01.2010
Chapter 2 Demand Filed: 03.11.2010
IPC:
C07D 495/04 (2006.01) ,A61K 31/4743 (2006.01) ,A61P 19/02 (2006.01) ,A61P 35/00 (2006.01) ,A61P 3/10 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
495
Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
02
in which the condensed system contains two hetero rings
04
Ortho-condensed systems
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
435
having six-membered rings with one nitrogen as the only ring hetero atom
47
Quinolines; Isoquinolines
4738
ortho- or peri-condensed with heterocyclic ring systems
4743
condensed with ring systems having sulfur as a ring hetero atom
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
19
Drugs for skeletal disorders
02
for joint disorders, e.g. arthritis, arthrosis
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
35
Antineoplastic agents
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
3
Drugs for disorders of the metabolism
08
for glucose homeostasis
10
for hyperglycaemia, e.g. antidiabetics
Applicants:
COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH [IN/IN]; Anusandhan Bhawan 2, Rafi Marg New Delhi 110 001, IN (AllExceptUS)
PANJAB UNIVERSITY [IN/IN]; Panjab University Chandigarh 160 014, IN (AllExceptUS)
KAKATIYA UNIVERSITY [IN/IN]; Kakatiya University Warangal 506 009, IN (AllExceptUS)
BOYAPATI, Shireesha [IN/IN]; IN (UsOnly)
RAO, Akkinepally, Raghuram [IN/IN]; IN (UsOnly)
NARSAIAH, Banda [IN/IN]; IN (UsOnly)
DIWAN, Prakash V. [IN/IN]; IN (UsOnly)
RAMAKRISHNA, Sistla [IN/IN]; IN (UsOnly)
MADHUSUDHANA [IN/IN]; IN (UsOnly)
YAKAIAH, Tallapally [IN/IN]; IN (UsOnly)
Inventors:
BOYAPATI, Shireesha; IN
RAO, Akkinepally, Raghuram; IN
NARSAIAH, Banda; IN
DIWAN, Prakash V.; IN
RAMAKRISHNA, Sistla; IN
MADHUSUDHANA; IN
YAKAIAH, Tallapally; IN
Agent:
SALHOTRA, Anuradha; LALL LAHIRI & SALHOTRA Plot No. B-28, Sector - 32 Institutional Area Gurgaon 122 001 Haryana, IN
Priority Data:
10/DEL/200905.01.2009IN
Title (EN) THIENOPYRIDINES AS PHARMACOLOGICALLY ACTIVE AGENTS
(FR) THIÉNOPYRIDINES SERVANT DE PRINCIPES ACTIFS PHARMACOLOGIQUES
Abstract:
(EN) The present invention provides compounds and pharmaceutically acceptable salts thereof methods for synthesizing thienopyridines and methods for inhibiting TNF- α activity for the treatment of cancer, asthma, arthritis, diabetes and inflammation. Provided- are compounds of formula (I).
(FR) L'invention concerne des composés de formule (I) et des sels pharmaceutiquement acceptables de ceux-ci, ainsi que des procédés pour synthétiser des thiénopyridines et des procédés pour inhiber l'activité du TNF-α pour le traitement du cancer, de l'asthme, de l'arthrite, du diabète et des inflammations.
front page image
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)
Also published as:
EP2373663JP2012514594US20110269790CN102341402CA2748982