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1. (WO2010075930) MODIFICATION I OF 4-({4-CARBOXYBUTYL)[2-(2-{[4-(2-PHENYLETHYL)BENZYL]OXY}PHENYL)ETHYL]-AMINO}METHYL)BENZOIC ACID
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2010/075930 International Application No.: PCT/EP2009/008664
Publication Date: 08.07.2010 International Filing Date: 04.12.2009
IPC:
C07C 229/38 (2006.01) ,A61K 31/197 (2006.01) ,A61P 9/00 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
229
Compounds containing amino and carboxyl groups bound to the same carbon skeleton
38
having amino groups bound to acyclic carbon atoms and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
185
Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
19
Carboxylic acids, e.g. valproic acid
195
having an amino group
197
the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid (GABA), beta-alanine, epsilon-aminocaproic acid, pantothenic acid
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
9
Drugs for disorders of the cardiovascular system
Applicants:
BAYER SCHERING PHARMA AKTIENGESELLSCHAFT [DE/DE]; Müllerstrasse 178 13353 Berlin, DE (AllExceptUS)
GRUNENBERG, Alfons [DE/DE]; DE (UsOnly)
MAIS, Franz-Josef [DE/DE]; DE (UsOnly)
TENBIEG, Katharina [DE/DE]; DE (UsOnly)
KEIL, Birgit [DE/DE]; DE (UsOnly)
Inventors:
GRUNENBERG, Alfons; DE
MAIS, Franz-Josef; DE
TENBIEG, Katharina; DE
KEIL, Birgit; DE
Common
Representative:
BAYER SCHERING PHARMA AKTIENGESELLSCHAFT [DE/DE]; Law and Patents Patents and Licensing 51368 Leverkusen, DE
Priority Data:
10 2008 062 689.917.12.2008DE
Title (DE) MODIFIKATION I DER 4-({4-CARBOXYBUTYL)[2-(2-{[4-(2-PHENYLETHYL)BENZYL]OXY}PHENYL)ETHYL]-AMINO}METHYL)BENZOESÄURE
(EN) MODIFICATION I OF 4-({4-CARBOXYBUTYL)[2-(2-{[4-(2-PHENYLETHYL)BENZYL]OXY}PHENYL)ETHYL]-AMINO}METHYL)BENZOIC ACID
(FR) MODIFICATION D'ACIDE 4-({4-CARBOXYBUTYL)[2-(2-{[4-(2-PHÉNYLÉTHYL)BENZYL]OXY}PHÉNYL)ÉTHYL]-AMINO}MÉTHYL)-BENZOÏQUE
Abstract:
(DE) Die Erfindung betrifft neue Formen der 4-({(4-Carboxybutyl)[2-(2-{[4-(2-phenylethyl)benzyl]oxy}phenyl)ethyl]amino}methyl)benzoesäure, insbesondere die Modifikation I, Verfahren zu deren Herstellung, diese enthaltende Arzneimittel sowie deren Verwendung bei der Bekämpfung von Krankheiten.
(EN) The invention relates to novel forms of 4-({(4-carboxybutyl)[2-(2-{[4-(2-phenylethyl)benzyl]oxy}phenyl)ethyl]amino}methyl)benzoic acid, especially modification I, methods for the production thereof, medicaments containing the same, and the use thereof for fighting diseases.
(FR) L'invention concerne de nouvelles formes d'acide 4-({4-carboxybutyl)[2-(2-{[4-(2-phényléthyl)benzyl]oxy}phényl)éthyl]-amino}méthyl)-benzoïque, notamment la modification I, des procédés de préparation de ces formes, des médicaments contenant ces formes et leur utilisation dans la lutte contre des maladies.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: German (DE)
Filing Language: German (DE)
Also published as:
AR075489EP2379489JP2012512204US20120010292CA2746870