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1. (WO2010075271) BICYCLIC HETEROCYCLE DERIVATIVES AND METHODS OF USE THEREOF
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2010/075271 International Application No.: PCT/US2009/068970
Publication Date: 01.07.2010 International Filing Date: 21.12.2009
IPC:
C07D 401/12 (2006.01) ,C07D 401/14 (2006.01) ,A61K 31/506 (2006.01) ,A61P 3/00 (2006.01) ,A61P 9/00 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
401
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
02
containing two hetero rings
12
linked by a chain containing hetero atoms as chain links
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
401
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
14
containing three or more hetero rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
495
having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
505
Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
506
not condensed and containing further heterocyclic rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
3
Drugs for disorders of the metabolism
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
9
Drugs for disorders of the cardiovascular system
Applicants:
SCHERING CORPORATION [US/US]; 126 East Lincoln Avenue RY60-30 Rahway, NJ 07065, US (AllExceptUS)
HARRIS, Joel M. [US/US]; US (UsOnly)
NEUSTADT, Bernard R. [US/US]; US (UsOnly)
STAMFORD, Andrew [AU/US]; US (UsOnly)
LIU, Hong [CN/US]; US (UsOnly)
Inventors:
HARRIS, Joel M.; US
NEUSTADT, Bernard R.; US
STAMFORD, Andrew; US
LIU, Hong; US
Agent:
BERGMAN, Jeffrey P.; Schering-Plough Corporation 2000 Galloping Hill Road Kenilworth, New Jersey 07033, US
Priority Data:
61/140,15623.12.2008US
Title (EN) BICYCLIC HETEROCYCLE DERIVATIVES AND METHODS OF USE THEREOF
(FR) DÉRIVÉS D'HÉTÉROCYCLES BICYCLIQUES ET LEURS PROCÉDÉS D'UTILISATION
Abstract:
(EN) The present invention relates to Bicyclic Heterocycle Derivatives, compositions comprising a Bicyclic Heterocycle Derivative, and methods of using the Bicyclic Heterocycle Derivatives for treating or preventing obesity, diabetes, a metabolic disorder, a cardiovascular disease or a disorder related to the activity of a GPCR in a patient.
(FR) La présente invention porte sur des dérivés d'hétérocycles bicycliques, sur des compositions comprenant un dérivé d'hétérocycle bicyclique et sur des procédés d'utilisation des dérivés d'hétérocycle bicyclique pour traiter ou prévenir l'obésité, le diabète, un trouble métabolique, une maladie cardiovasculaire ou un trouble lié à l'activité d'un RCPG chez un patient.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)
Also published as:
EP2382203JP2012513470US20110263624CA2747809AU2009330208