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1. (WO2010072754) HYDROSOLUBLE [6)O-α-D-GLCP-(1→]n-6-O-β-D-GLCP-(1→-PHENOLIC DERIVATIVES WITH DERMOCOSMETIC, NUTRITIONAL AND THERAPEUTIC APPLICATIONS, AND COMPOSITIONS CONTAINING SAID WATER SOLUBLE COMPOUNDS
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2010/072754 International Application No.: PCT/EP2009/067736
Publication Date: 01.07.2010 International Filing Date: 22.12.2009
IPC:
C07H 15/203 (2006.01) ,C07H 15/26 (2006.01) ,A61K 8/00 (2006.01) ,A61K 31/7034 (2006.01) ,A61P 35/00 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
H
SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
15
Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
20
Carbocyclic rings
203
Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
H
SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
15
Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
26
Acyclic or carbocyclic radicals, substituted by hetero rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
8
Cosmetics or similar toilet preparations
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
70
Carbohydrates; Sugars; Derivatives thereof
7028
Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
7034
attached to a carbocyclic compound, e.g. phloridzin
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
35
Antineoplastic agents
Applicants:
LIBRAGEN [FR/FR]; 3 rue des Satellites Bât. Canal Biotech F-31000 Toulouse, FR (AllExceptUS)
AURIOL, Daniel [FR/FR]; FR (UsOnly)
GINOLHAC, Aurélien [FR/FR]; FR (UsOnly)
LEFEVRE, Fabrice [FR/FR]; FR (UsOnly)
NALIN, Renaud [FR/FR]; FR (UsOnly)
Inventors:
AURIOL, Daniel; FR
GINOLHAC, Aurélien; FR
LEFEVRE, Fabrice; FR
NALIN, Renaud; FR
Agent:
GALLOIS, Valérie; Becker & Associés 25 rue Louis Le Grand F-75002 Paris, FR
Priority Data:
08306007.923.12.2008EP
Title (EN) HYDROSOLUBLE [6)O-α-D-GLCP-(1→]n-6-O-β-D-GLCP-(1→-PHENOLIC DERIVATIVES WITH DERMOCOSMETIC, NUTRITIONAL AND THERAPEUTIC APPLICATIONS, AND COMPOSITIONS CONTAINING SAID WATER SOLUBLE COMPOUNDS
(FR) DÉRIVÉS [6)-0-Α-D-GLCP-(1→]N-6-O-Β-D-GLCP-(1→-PHÉNOLIQUES POUR APPLICATIONS DERMOCOSMÉTIQUES, ALIMENTAIRES ET THÉRAPEUTIQUES, ET COMPOSITIONS CONTENANT LESDITS COMPOSÉS HYDROSOLUBLES
Abstract:
(EN) The invention relates to [6)-O-α-D-Glcp→]1 →]n-6-O-β-D-Glcp-(1→-phenolic derivatives. These [6)-O-α-D-Glcp-(1→]n-6-O-β-D-Glcp-(1→-phenolic derivatives of selected phenolics are new, have a solubility in water higher than that of their parent O-β-D-Glcp- (1→-phenolic derivatives and have useful applications in cosmetic, nutrition and pharmaceutical compositions, such as treating or preventing oxidative stress, a cancer, a cardiovascular disease, a bacterial infection, a viral infection, a fungal infection, a UV- induced erythema, an allergy, a metabolism disorder, diabetes, an obesity, an hormonal disorder, a bone disease, a pain, a brain disease, a mouth or teeth disease, an inflammatory or immune disorder.
(FR) La présente invention concerne de nouveaux dérivés [6)-0-α-D-Glcp-(1→]n-6-O-β-D-Glcp-(1→-phénoliques dont la solubilité dans l'eau est supérieure à celle de leurs dérivés O-β-D-Glcp-(1→-phénoliques parents et qui possèdent des applications utiles dans des compositions cosmétiques, alimentaires et pharmaceutiques, par exemple pour le traitement ou la prévention du stress oxydatif, d'un cancer, d'une maladie cardiovasculaire, d'une infection bactérienne, virale ou fongique, d'un érythème induit par les UV, d'une allergie, d'un trouble métabolique, du diabète, de l'obésité, d'un trouble hormonal, d'une maladie des os, d'une douleur, d'une maladie cérébrale, d'une maladie de la bouche ou des dents, d'un trouble inflammatoire ou d'un trouble immunitaire.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)
Also published as:
EP2379576US20110256115KR1020110106415