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1. (WO2010072742) PROCESSES AND INTERMEDIATES FOR PREPARING A MACROCYCLIC PROTEASE INHIBITOR OF HCV
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2010/072742 International Application No.: PCT/EP2009/067715
Publication Date: 01.07.2010 International Filing Date: 22.12.2009
IPC:
C07D 311/06 (2006.01) ,C07D 417/04 (2006.01) ,C07D 453/04 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
311
Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
02
ortho- or peri-condensed with carbocyclic rings or ring systems
04
Benzo [b] pyrans, not hydrogenated in the carbocyclic ring
06
with oxygen or sulfur atoms directly attached in position 2
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
417
Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/196
02
containing two hetero rings
04
directly linked by a ring-member-to-ring- member bond
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
453
Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
02
containing not further condensed quinuclidine ring systems
04
having a quinolyl-4, a substituted quinolyl-4 or a alkylenedioxy-quinolyl-4 radical linked through only one carbon atom, attached in position 2, e.g. quinine
Applicants:
ORTHO-MCNEIL-JANSSEN PHARMACEUTICALS, Inc [US/US]; 1125 Trenton-Harbourton Road Titusville, New Jersey 08560, US (AllExceptUS)
HORVATH, Andras [HU/BE]; BE (UsOnly)
ORMEROD, Dominic John [GB/BE]; BE (UsOnly)
DEPRÉ, Dominique Paul Michel [BE/BE]; BE (UsOnly)
CERPENTIER, Véronique [BE/BE]; BE (UsOnly)
Inventors:
HORVATH, Andras; BE
ORMEROD, Dominic John; BE
DEPRÉ, Dominique Paul Michel; BE
CERPENTIER, Véronique; BE
Agent:
WANTE, Dirk; Tibotec-Virco Comm. VA J&J Patent Law Department Generaal De Wittelaan L 11B 3 B-2800 Mechelen, BE
Priority Data:
08172691.123.12.2008EP
Title (EN) PROCESSES AND INTERMEDIATES FOR PREPARING A MACROCYCLIC PROTEASE INHIBITOR OF HCV
(FR) PROCÉDÉS ET INTERMÉDIAIRES POUR PRÉPARER UN INHIBITEUR MACROCYCLIQUE DE PROTÉASE DU VHC
Abstract:
(EN) The present invention relates to the cinchonidine salt useful in the preparation of intermediates for preparing a macrocyclic HCV inhibitor, as well as processes involving this salt.
(FR) La présente invention porte sur le sel de cinchonidine utile dans la préparation d'intermédiaires pour préparer un inhibiteur macrocyclique du VHC ainsi que sur des procédés utilisant ce sel.
front page image
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)
Also published as:
AR074863IL213246MXMX/a/2011/006764EP2382198JP2012513381US20110257403
CN102264715RU2011130895CA2745565ES2429013PT2382198MX2011006764
US20150080577KR1020110099048BRPI0923393RU0002588132DK2382198AU2009331530
IN1505/MUMNP/2011RU2016120007