Search International and National Patent Collections
Some content of this application is unavailable at the moment.
If this situation persists, please contact us atFeedback&Contact
1. (WO2010072354) MESYLATE SALT OF 5-(2-{[6-(2,2-DIFLUORO-2-PHENYLETHOXY)HEXYL]AMINO }-1-HYDROXYETHYL)-8-HYDROXYQUINOLIN-2(1H)-ONE AS AGONIST OF THE β2 ADRENERGIC RECEPTOR
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2010/072354 International Application No.: PCT/EP2009/008970
Publication Date: 01.07.2010 International Filing Date: 15.12.2009
IPC:
C07D 215/26 (2006.01) ,A61K 31/4704 (2006.01) ,A61P 11/00 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
215
Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
02
having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
16
with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
20
Oxygen atoms
24
attached in position 8
26
Alcohols; Ethers thereof
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
435
having six-membered rings with one nitrogen as the only ring hetero atom
47
Quinolines; Isoquinolines
4704
2-Quinolinones, e.g. carbostyril
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
11
Drugs for disorders of the respiratory system
Applicants:
ALMIRALL, S.A. [ES/ES]; Ronda del General Mitre 151 E-08022 Barcelona, ES (AllExceptUS)
CARRERA CARRERA, Francesc [ES/ES]; ES (UsOnly)
PUIG DURAN, Carlos [ES/ES]; ES (UsOnly)
MARCHUETA HEREU, Iolanda [ES/ES]; ES (UsOnly)
MOYES VALLS, Enrique [ES/ES]; ES (UsOnly)
Inventors:
CARRERA CARRERA, Francesc; ES
PUIG DURAN, Carlos; ES
MARCHUETA HEREU, Iolanda; ES
MOYES VALLS, Enrique; ES
Agent:
SRINIVASAN, Ravi Chandran; J.A. Kemp & Co. 14 South Square, Gray's Inn London WC1R 5JJ, GB
Priority Data:
08382082.922.12.2008EP
Title (EN) MESYLATE SALT OF 5-(2-{[6-(2,2-DIFLUORO-2-PHENYLETHOXY)HEXYL]AMINO }-1-HYDROXYETHYL)-8-HYDROXYQUINOLIN-2(1H)-ONE AS AGONIST OF THE β2 ADRENERGIC RECEPTOR
(FR) SEL DE MÉSYLATE DE 5-(2-{[6-(2,2-DIFLUORO-2-PHÉNYLÉTHOXY)HEXYL]AMINO }-1-HYDROXYÉTHYL)-8-HYDROXYQUINOLÉIN-2(1H)-ONE COMME AGONISTE DU RÉCEPTEUR Β2 ADRÉNERGIQUE
Abstract:
(EN) The present invention is directed to a mesylate salt of 5-(2-{[6-(2,2-difluoro-2- phenylethoxy)hexyl]amino}-1-hydroxyethyl)-8-hydroxyquinolin-2(1 H)-one and pharmaceutically acceptable solvates thereof.
(FR) La présente invention a pour objet un sel de mésylate de 5-(2-{[6-(2,2-difluoro-2- phényléthoxy)hexyl]amino}-1-hydroxyéthyl)-8-hydroxyquinoléin-2(1 H)-one et des solvates pharmaceutiquement acceptables de celui-ci.
front page image
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)
Also published as:
RSP-2012/0554UAa201109111UY0001032297AR074792IL213161EP2367796
MXMX/a/2011/006491SG171992JP2012513424US20110251234ES2397209CN102264703
CA2748105EA201100970PT2367796MX2011006491CO6390056CL2011001544
KR1020110103397NZ592797AU2009331961VN28540ID051.4342MYPI 2011002871
TH127128BRPI0918370IN4776/DELNP/2011