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1. (WO2010030704) ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2010/030704    International Application No.:    PCT/US2009/056407
Publication Date: 18.03.2010 International Filing Date: 09.09.2009
IPC:
C07H 15/232 (2006.01), A61K 31/704 (2006.01), A61P 31/04 (2006.01)
Applicants: ACHAOGEN, INC. [US/US]; 7000 Shoreline Court, 3rd Floor South San Francisco, California 94080 (US) (For All Designated States Except US).
AGGEN, James, Bradley [US/US]; (US) (For US Only).
LINSELL, Martin, Sheringham [GB/US]; (US) (For US Only).
GOLDBLUM, Adam, Aaron [US/US]; (US) (For US Only).
HILDEBRANDT, Darin, James [US/US]; (US) (For US Only).
KANE, Timothy, Robert [US/US]; (US) (For US Only).
DOZZO, Paola [IT/US]; (US) (For US Only).
GLIEDT, Micah, James [US/US]; (US) (For US Only).
HANESSIAN, Stephen [US/CA]; (CA) (For US Only).
GIGUERE, Alexandre [CA/CA]; (CA) (For US Only).
GRZYB, Justyna [CA/CA]; (CA) (For US Only).
MAIANTI, Juan, Pablo [UY/CA]; (CA) (For US Only)
Inventors: AGGEN, James, Bradley; (US).
LINSELL, Martin, Sheringham; (US).
GOLDBLUM, Adam, Aaron; (US).
HILDEBRANDT, Darin, James; (US).
KANE, Timothy, Robert; (US).
DOZZO, Paola; (US).
GLIEDT, Micah, James; (US).
HANESSIAN, Stephen; (CA).
GIGUERE, Alexandre; (CA).
GRZYB, Justyna; (CA).
MAIANTI, Juan, Pablo; (CA)
Agent: WAGNER, Emily, W.; Seed Intellectual Property Law Group PLLC Suite 5400 701 Fifth Avenue Seattle, Washington 98104-7064 (US)
Priority Data:
61/095,673 10.09.2008 US
Title (EN) ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS
(FR) ANALOGUES D’AMINOGLYCOSIDES ANTIBACTÉRIENS
Abstract: front page image
(EN)Compounds having antibacterial activity are disclosed. The compounds have the following structure (I) including stereoisomers, pharmaceutically acceptable salts and prodrugs thereof, wherein Q1, Q2, Z1, Z2, Z3, Z4, R1, R2 and R3 are as defined herein. Methods associated with preparation and use of such compounds, as well as pharmaceutical compositions comprising such compounds, are also disclosed.
(FR)La présente invention concerne des composés possédant une activité antimicrobienne. Les composés possèdent la structure (I) suivante : y compris ses stéréoisomères, ses sels acceptables sur le plan pharmaceutique et ses promédicaments, où Q1, Q2, Z1, Z2, Z3, Z4, R1, R2 et R3 sont tels que définis ci-dessus. Des procédés associés à la préparation et à l’utilisation de ces composés, ainsi que des compositions pharmaceutiques contenant ces composés, sont également décrits.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)