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1. (WO2010029938) NOVEL CRYSTAL FORMS OF 4-(2-AMINOPYRIDIN-4-YL)-3-(4–FLUORO- PHENYL)-1-(1,4,5,6-TETRAHYDRO-6-OXOPYRIDAZIN-3-YL)-1H-PYRA-ZOLE METHANESULFONATE AND PROCESS FOR PRODUCTION OF SAME
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2010/029938    International Application No.:    PCT/JP2009/065728
Publication Date: 18.03.2010 International Filing Date: 09.09.2009
IPC:
C07D 401/14 (2006.01), A61K 31/501 (2006.01), A61P 19/02 (2006.01), A61P 29/00 (2006.01), A61P 43/00 (2006.01)
Applicants: UBE INDUSTRIES, LTD. [JP/JP]; 1978-96, Oaza Kogushi, Ube-shi, Yamaguchi 7558633 (JP) (For All Designated States Except US).
SHIMIZU, Motohisa; (For US Only).
SUZUKI, Naoto; (For US Only).
MOTOYAMA, Takahiro; (For US Only).
MIYATA, Hiroyuki; (For US Only)
Inventors: SHIMIZU, Motohisa; .
SUZUKI, Naoto; .
MOTOYAMA, Takahiro; .
MIYATA, Hiroyuki;
Agent: TSUKUNI, Hajime; KASUMIGASEKI TOKYU Bldg., 3-7-1, Kasumigaseki, Chiyoda-ku, Tokyo 1000013 (JP)
Priority Data:
2008-230898 09.09.2008 JP
Title (EN) NOVEL CRYSTAL FORMS OF 4-(2-AMINOPYRIDIN-4-YL)-3-(4–FLUORO- PHENYL)-1-(1,4,5,6-TETRAHYDRO-6-OXOPYRIDAZIN-3-YL)-1H-PYRA-ZOLE METHANESULFONATE AND PROCESS FOR PRODUCTION OF SAME
(FR) NOUVELLES FORMES CRISTALLINES DE 4-(2-AMINOPYRIDIN-4-YL)-3-(4–FLUORO- PHÉNYL)-1-(1,4,5,6-TÉTRAHYDRO-6-OXOPYRIDAZIN-3-YL)-1H-PYRAZOLE-MÉTHANESULFONATE ET PROCÉDÉ POUR LA PRODUCTION DE CELLES-CI
(JA) 4-(2-アミノピリジン-4-イル)-3-(4-フルオロフェニル)-1-(1,4,5,6-テトラヒドロ-6-オキソピリダジン-3-イル)-1H-ピラゾール メタンスルホン酸塩の新規結晶形及びその製造方法
Abstract: front page image
(EN)Novel crystal forms of 4-(2-aminopyridin-4-yl)-3-(4- fluorophenyl)-1-(1,4,5,6-tetrahydro-6-oxopyridazin-3-yl)-1H-pyrazole methanesulfonate, which are useful as medicines; and a process for production of same. Two stable polymorphic forms called A-type crystal and B-type crystal; and a process for production by which the polymorphic forms can be each produced as a single polymorphic form.
(FR)La présente invention concerne de nouvelles formes cristallines de 4-(2-aminopyridin-4-yl)-3-(4-fluorophényl)-1-(1,4,5,6-tétrahydro-6-oxopyridazin-3-yl)-1H-pyrazole-méthanesulfonate, qui sont utiles en tant que médicaments; et un procédé pour la production de celles-ci. Deux formes polymorphes stables appelées cristal de type A et cristal de type B; et un procédé de production par lequel chacune des formes polymorphes peut être produite sous la forme d'une forme polymorphe unique.
(JA) 本発明は、医薬品として有用な、4-(2-アミノピリジン-4-イル)-3-(4-フルオロフェニル)-1-(1,4,5,6-テトラヒドロ-6-オキソピリダジン-3-イル)-1H-ピラゾール メタンスルホン酸塩の新規結晶形及びその製造方法に関する。 本発明は、A型結晶及びB型結晶と称される安定な2つの結晶多形と、かかる結晶多形をそれぞれ単一の結晶として得ることができる製造方法とを提供する。
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: Japanese (JA)
Filing Language: Japanese (JA)