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1. (WO2010028033) AMIDES OF DIAZABICYCLOOCTANES AND USES THEREOF
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2010/028033    International Application No.:    PCT/US2009/055718
Publication Date: 11.03.2010 International Filing Date: 02.09.2009
IPC:
C07D 471/08 (2006.01), A61K 31/407 (2006.01), A61P 25/00 (2006.01)
Applicants: TARGACEPT, INC. [US/US]; 200 East First Street, Suite 300 Winston-Salem, North Carolina 27101 (US) (For All Designated States Except US).
STRACHAN, Jon-Paul [GB/US]; (US) (For US Only).
BHATTI, Balwinder Singh [US/US]; (US) (For US Only).
MAZUROV, Anatoly [US/US]; (US) (For US Only).
KLUCIK, Jozef [US/US]; (US) (For US Only).
XIAO, Yun-De [CN/US]; (US) (For US Only).
HAMMOND, Philip S. [US/US]; (US) (For US Only).
KOMBO, David [CG/US]; (US) (For US Only).
MIAO, Lan [US/US]; (US) (For US Only).
SPEAKE, Jason Daniel [US/US]; (US) (For US Only).
YOHANNES, Daniel [ER/US]; (US) (For US Only)
Inventors: STRACHAN, Jon-Paul; (US).
BHATTI, Balwinder Singh; (US).
MAZUROV, Anatoly; (US).
KLUCIK, Jozef; (US).
XIAO, Yun-De; (US).
HAMMOND, Philip S.; (US).
KOMBO, David; (US).
MIAO, Lan; (US).
SPEAKE, Jason Daniel; (US).
YOHANNES, Daniel; (US)
Agent: FIX, Amy H.; (US)
Priority Data:
61/094,647 05.09.2008 US
Title (EN) AMIDES OF DIAZABICYCLOOCTANES AND USES THEREOF
(FR) AMIDES DE DIAZABICYCLOOCTANES ET LEURS UTILISATIONS
Abstract: front page image
(EN)The present invention relates to compounds of the following formulae I and II that bind to and modulate the activity of neuronal nicotinic acetylcholine receptors, to processes for preparing these compounds, to pharmaceutical compositions containing these compounds, and to methods of using these compounds for treating a wide variety of conditions and disorders, including those associated with dysfunction of the central nervous system (CNS). Formula (I ), Formula (Il)
(FR)La présente invention porte sur des composés représentés par les formules I et II suivantes, qui se lient à et modulent l'activité de récepteurs nicotiniques neuronaux de l'acétylcholine, sur des procédés de préparation de ces composés, sur des compositions pharmaceutiques contenant ces composés, et sur des méthodes d'utilisation de ces composés pour le traitement d'une large diversité d'états pathologiques et de troubles, comprenant ceux associés à un dysfonctionnement du système nerveux central (CNS).
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)