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1. (WO2010027510) ENANTIOSELECTIVE CASCADE MICHAEL-MICHAEL REACTIONS AND RELATED CATALYSTS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2010/027510    International Application No.:    PCT/US2009/005042
Publication Date: 11.03.2010 International Filing Date: 08.09.2009
IPC:
C07D 207/335 (2006.01), C07D 207/337 (2006.01), C07D 207/12 (2006.01), C07D 207/10 (2006.01)
Applicants: STC. UNM [US/US]; 801 University Blvd. SE, Suite 101 Albuquerque, NM 87106 (US) (For All Designated States Except US).
WANG, Wei [CN/US]; (US) (For US Only)
Inventors: WANG, Wei; (US)
Agent: COLEMAN, Henry, D.; (US)
Priority Data:
61/191,486 08.09.2008 US
Title (EN) ENANTIOSELECTIVE CASCADE MICHAEL-MICHAEL REACTIONS AND RELATED CATALYSTS
(FR) RÉACTIONS DE DOUBLE MICHAËL ÉNANTIOSÉLECTIVES EN CASCADE ET CATALYSEURS ASSOCIÉS
Abstract: front page image
(EN)The invention provides direct processes and related catalysts for the syntheses of trisubstituted chiral pyrrolidines, piperidines, tetrahydrothiophenes, and thianes by highly enantio- and diastereoselective cascade Michael-Michael reaction of α, β-unsaturatedaldehydes with /ra/25-γ-protected amino α, β-unsaturated esters.
(FR)La présente invention concerne des procédés directs et des catalyseurs associés pour les synthèses de pyrrolidines chirales trisubstituées, de pipéridines, de tétrahydrothiophènes, et de thianes par la réaction de Double Michaël énantio- et diastéréosélective en cascade d’aldéhydes α,β-insaturés avec des amino esters α, β-insaturés /ra/25-γ-protégés.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)