Processing

Please wait...

Settings

Settings

Goto Application

1. WO2010003702 - SYNTHESIS OF PALIPERIDONE

Publication Number WO/2010/003702
Publication Date 14.01.2010
International Application No. PCT/EP2009/005099
International Filing Date 10.07.2009
IPC
C07D 471/04 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
471Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/-C07D463/251
02in which the condensed system contains two hetero rings
04Ortho-condensed systems
CPC
C07D 471/04
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
471Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
02in which the condensed system contains two hetero rings
04Ortho-condensed systems
Applicants
  • SYNTHON B.V. [NL]/[NL] (AllExceptUS)
  • BARTL, Jiri [CZ]/[CZ] (UsOnly)
  • BENOVSKY, Petr [CZ]/[CZ] (UsOnly)
Inventors
  • BARTL, Jiri
  • BENOVSKY, Petr
Agents
  • PRINS, Hendrik, Willem
Priority Data
61/080,07211.07.2008US
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) SYNTHESIS OF PALIPERIDONE
(FR) SYNTHÈSE DE PALIPÉRIDONE
Abstract
(EN)
A compound of formula (6) or an acid addition salt thereof in which G is (i) a leaving group A selected from a halo group and a sulfonyloxy group, or (ii) a group of the formula (20) is useful in processes of making paliperidone and related compounds.
(FR)
La présente invention concerne un composé de formule (6) ou un sel d'addition aux acides de celui-ci dans lequel G est (i) un groupe partant choisi parmi un groupe halogéno et un groupe sulfonyloxy, ou (ii) un groupe de formule (20) et qui est utile dans les procédés de fabrication de palipéridone et composés associés.
Also published as
Latest bibliographic data on file with the International Bureau