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1. (WO2009139181) 10A-AZALIDE COMPOUND HAVING 4-MEMBERED RING STRUCTURE
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2009/139181    International Application No.:    PCT/JP2009/002135
Publication Date: 19.11.2009 International Filing Date: 15.05.2009
IPC:
C07H 17/00 (2006.01), A61K 31/7052 (2006.01), A61P 31/04 (2006.01)
Applicants: TAISHO PHARMACEUTICAL CO., LTD. [JP/JP]; 24-1, Takada 3-chome, Toshima-ku, Tokyo 1708633 (JP) (For All Designated States Except US).
MEIJI SEIKA KAISHA, LTD. [JP/JP]; 4-16, Kyobashi 2-chome, Chuo-ku, Tokyo 1048002 (JP) (For All Designated States Except US).
SUGIMOTO, Tomohiro [JP/JP]; (JP) (For US Only).
YAMAMOTO, Kanako [JP/JP]; (JP) (For US Only).
KUROSAKA, Jun [JP/JP]; (JP) (For US Only).
SASAMOTO, Naoki [JP/JP]; (JP) (For US Only).
KASHIMURA, Masato [JP/JP]; (JP) (For US Only).
MIURA, Tomoaki [JP/JP]; (JP) (For US Only).
KANEMOTO, Kenichi [JP/JP]; (JP) (For US Only).
YOSHIDA, Satoshi [JP/JP]; (JP) (For US Only).
KUMURA, Kou [JP/JP]; (JP) (For US Only).
AJITO, Keiichi [JP/JP]; (JP) (For US Only)
Inventors: SUGIMOTO, Tomohiro; (JP).
YAMAMOTO, Kanako; (JP).
KUROSAKA, Jun; (JP).
SASAMOTO, Naoki; (JP).
KASHIMURA, Masato; (JP).
MIURA, Tomoaki; (JP).
KANEMOTO, Kenichi; (JP).
YOSHIDA, Satoshi; (JP).
KUMURA, Kou; (JP).
AJITO, Keiichi; (JP)
Agent: SIKs & Co.; 8th Floor, Kyobashi-Nisshoku Bldg., 8-7, Kyobashi 1-chome, Chuo-ku, Tokyo 1040031 (JP)
Priority Data:
2008-127832 15.05.2008 JP
2009-024457 05.02.2009 JP
Title (EN) 10A-AZALIDE COMPOUND HAVING 4-MEMBERED RING STRUCTURE
(FR) COMPOSÉ 10A-AZALIDE AYANT UNE STRUCTURE DE CYCLE À 4 CHAÎNONS
(JA) 4員環構造を有する10a-アザライド化合物
Abstract: front page image
(EN)Disclosed is a 10a-azalide compound which is effective against a bacterium Haemophilus influenzae (an influenza bacterium) or an erythromycin-resistant bacterium (e.g., resistant pneumococcus or streptococcus) and has a novel structure.  The 10a-azalide compound is represented by formula (I) and has a 4-membered ring structure cross-linked at position-10a and position-12.
(FR)La présente invention concerne un composé 10a-azalide qui est efficace contre une bactérie Haemophilus influenzae (une bactérie influenza) ou une bactérie résistant à l'érythromycine (par exemple, un pneumocoque ou un streptocoque résistant) et présente une nouvelle structure. Le composé 10a-azalide est représenté par la formule (I) et a une structure de cycle à 4 chaînons réticulé en position 10a et en position 12.
(JA) インフルエンザ菌又はエリスロマイシン耐性菌(例えば耐性肺炎球菌及び連鎖球菌)に対しても有効な新規構造を有する式(I)で表される10a及び12位で架橋された4員環構造を有する10a-アザライド化合物。
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: Japanese (JA)
Filing Language: Japanese (JA)