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Machine translation
1. (WO2009135526) ALPHA-MERCAPTO-AMIDES
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2009/135526    International Application No.:    PCT/EP2008/055594
Publication Date: 12.11.2009 International Filing Date: 07.05.2008
IPC:
C07C 323/60 (2006.01), C07D 231/40 (2006.01), C07D 241/20 (2006.01), C07D 263/56 (2006.01), C07D 277/64 (2006.01), C07D 285/135 (2006.01), A61K 31/16 (2006.01), A61K 31/165 (2006.01), A61K 31/415 (2006.01), A61K 31/423 (2006.01), A61K 31/428 (2006.01), A61K 31/433 (2006.01), A61K 31/53 (2006.01), A61P 3/04 (2006.01), A61P 3/10 (2006.01)
Applicants: NOVARTIS AG [CH/CH]; Lichtstrasse 35 CH-4056 Basel (CH) (For All Designated States Except US).
NAPOLETANO, Mauro [IT/IT]; (IT) (For US Only).
HAACK, Thomas [DE/IT]; (IT) (For US Only).
TSCHINKE, Vincenzo [IT/CH]; (CH) (For US Only).
JELAKOVIC, Stjepan [HR/DE]; (DE) (For US Only).
MAH, Robert [CA/CH]; (CH) (For US Only)
Inventors: NAPOLETANO, Mauro; (IT).
HAACK, Thomas; (IT).
TSCHINKE, Vincenzo; (CH).
JELAKOVIC, Stjepan; (DE).
MAH, Robert; (CH)
Priority Data:
Title (EN) ALPHA-MERCAPTO-AMIDES
(FR) ALPHA-MERCAPTOAMIDES
Abstract: front page image
(EN)Substituted amides of the general formula (I): with the residues A, R1 and R2 as explained in detail in the description are described. The compounds are suitable in particular as neutral endopeptidase inhibitors and are highly potent.
(FR)L'invention porte sur des amides substitués représentés par la formule générale (I), dans laquelle les résidus A, R1 et R2 sont tels qu'expliqués en détail dans la description. Les composés sont très puissants et sont appropriés en particulier comme inhibiteurs de l'endopeptidase neutre.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MT, NL, NO, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)