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Machine translation
1. (WO2009129259) POLYMORPHS OF 5-(3-(ETHYLSULFONYL)PHENYL)-3,8-DIMETHYL-N-(1-METHYLPIPERIDIN-4-YL)-9H-PYRIDO[2,3-B]INDOLE-7-CARBOXAMIDE AND METHODS OF USE THEREFOR
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2009/129259    International Application No.:    PCT/US2009/040556
Publication Date: 22.10.2009 International Filing Date: 14.04.2009
IPC:
C07D 471/04 (2006.01), A61K 31/437 (2006.01), A61P 35/00 (2006.01), A61P 25/00 (2006.01)
Applicants: TAKEDA PHARMACEUTICAL COMPANY LIMITED [JP/JP]; 1-1 Doshomachi, 4-come, Chuo-ku Osaka-shi , Osaka, 541-0045 (JP) (For All Designated States Except US).
ISBESTER, Paul [US/US]; (US) (For US Only).
PALMER, Grant, J. [US/US]; (US) (For US Only).
MOBELE, Bingidimi, I. [CD/US]; (US) (For US Only).
SALSBURY, Jonathon, S. [US/US]; (US) (For US Only).
ULYSEE, Luckner [US/US]; (US) (For US Only)
Inventors: ISBESTER, Paul; (US).
PALMER, Grant, J.; (US).
MOBELE, Bingidimi, I.; (US).
SALSBURY, Jonathon, S.; (US).
ULYSEE, Luckner; (US)
Agent: SMITH, C. Amy; (US)
Priority Data:
61/045,458 16.04.2008 US
Title (EN) POLYMORPHS OF 5-(3-(ETHYLSULFONYL)PHENYL)-3,8-DIMETHYL-N-(1-METHYLPIPERIDIN-4-YL)-9H-PYRIDO[2,3-B]INDOLE-7-CARBOXAMIDE AND METHODS OF USE THEREFOR
(FR) POLYMORPHES DE 5-(3-(ÉTHYLSULFONYL)PHÉNYL)-3,8-DIMÉTHYL-N-(1-MÉTHYLPIPÉRIDIN-4-YL)-9H-PYRIDO[2,3-B]INDOLE-7-CARBOXAMIDE ET PROCÉDÉS D'UTILISATION ASSOCIÉS
Abstract: front page image
(EN)The invention relates to polymorphic forms of 5-(3-(ethylsulfonyl)phenyl)-3,8-dimethyl-N-(1-methylpiperidin-4-yl)-9h-pyrido[2,3-b]indole-7-carboxamide (referred to herein as Compound I), which has the formula: (A). The invention also relates to compositions thereof and methods for the preparation of the polymorphs of Compound I, and kits and articles of manufacture of the compositions, and methods of using the compositions to treat various diseases.
(FR)L'invention concerne des formes polymorphes de 5-(3-(éthylsulfonyl)phényl)-3,8-diméthyl-N-(1-méthylpipéridin-4-yl)-9h-pyrido[2,3-b]indole-7-carboxamide (appelé ci-après composé I), ce composé étant représenté par la formule: ##STR##. L'invention concerne aussi des compositions de celui-ci et des procédés de préparation des polymorphes du composé I, ainsi que des trousses et des articles fabriqués à l'aide de ces compositions et des procédés d'utilisation de ces compositions pour traiter diverses maladies.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)