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1. (WO2009127623) CRYSTALLINE (6R,7R)-7-{2-(5-AMINO-[1,2,4]THIADIAZOL-3-YL)-2-[(Z)-TRITYLOXYIMINO]-ACETYLAMINO}-3-[(R)-1'-TERT-BUTOXYCARBONYL-2-OXO-[1,3']BIPYRROLIDINYL-(3E)-YLIDENEMETHYL]-8-OXO-5-THIA-1-AZA-BICYCLO[4.2.0]OCT-2-ENE-2-CARBOXYLIC ACID BENZHYDRYL ESTER; ITS MANUFACTURE AND USE
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2009/127623    International Application No.:    PCT/EP2009/054405
Publication Date: 22.10.2009 International Filing Date: 14.04.2009
IPC:
C07D 501/12 (2006.01), C07D 501/54 (2006.01), A61P 31/00 (2006.01), A61K 31/546 (2006.01)
Applicants: BASILEA PHARMACEUTICA AG [CH/CH]; Grenzacherstrasse 487 CH-4005 Basel (CH) (For All Designated States Except US).
ALPEGIANI, Marco [IT/IT]; (IT) (For US Only).
CABRI, Walter [IT/IT]; (IT) (For US Only).
HEUBES, Markus [DE/DE]; (DE) (For US Only).
LONGONI, Davide [IT/IT]; (IT) (For US Only).
SCHLEIMER, Michael [DE/DE]; (DE) (For US Only)
Inventors: ALPEGIANI, Marco; (IT).
CABRI, Walter; (IT).
HEUBES, Markus; (DE).
LONGONI, Davide; (IT).
SCHLEIMER, Michael; (DE)
Agent: BOHEST AG; P.O. Box 160 CH-4003 Basel (CH)
Priority Data:
08154517.0 15.04.2008 EP
Title (EN) CRYSTALLINE (6R,7R)-7-{2-(5-AMINO-[1,2,4]THIADIAZOL-3-YL)-2-[(Z)-TRITYLOXYIMINO]-ACETYLAMINO}-3-[(R)-1'-TERT-BUTOXYCARBONYL-2-OXO-[1,3']BIPYRROLIDINYL-(3E)-YLIDENEMETHYL]-8-OXO-5-THIA-1-AZA-BICYCLO[4.2.0]OCT-2-ENE-2-CARBOXYLIC ACID BENZHYDRYL ESTER; ITS MANUFACTURE AND USE
(FR) ESTER BENZHYDRYLIQUE DE L'ACIDE (6R,7R)-7-{2-(5-AMINO-[1,2,4]THIADIAZOL-3-YL)-2-[(Z)-TRITYLOXYIMINO]-ACÉTYLAMINO}-3-[(R)-1'-TERT-BUTOXYCARBONYL-2-OXO-[1,3']BIPYRROLIDINYL-(3E)-YLIDÈNEMÉTHYL]-8-OXO-5-THIA-1-AZA-BICYCLO[4.2.0]OCT-2-ÈNE-2-CARBOXYLIQUE CRISTALLIN ; SA FABRICATION ET SON UTILISATION
Abstract: front page image
(EN)A solid DMSO solvate of a compound of formula (I) is described, which is a useful intermediate for preparing the broad spectrum antibiotics Ceftobiprole and Ceftobiprole Medocaril.
(FR)L'invention porte sur un solvate avec le DMSO solide d'un composé de formule (I), qui est un intermédiaire utile pour la préparation des antibiotiques à large spectre Ceftobiprole et Ceftobiprole Medocaril.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)