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1. WO2009115393 - PROCESS FOR THE PREPARATION OF N-(1-PHENYLETHYL)ANILINES, SALTS, AND SOLVATES THEREOF USEFUL AS SEROTONIN 5-HT6 ANTAGONISTS

Publication Number WO/2009/115393
Publication Date 24.09.2009
International Application No. PCT/EP2009/052066
International Filing Date 20.02.2009
IPC
C07C 211/00 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
211Compounds containing amino groups bound to a carbon skeleton
C07D 295/00 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
295Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
C07C 251/00 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
251Compounds containing nitrogen atoms doubly- bound to a carbon skeleton
CPC
C07C 317/40
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
317Sulfones; Sulfoxides
26having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
32with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
34having sulfone or sulfoxide groups and amino groups bound to carbon atoms of six-membered aromatic rings being part of the same non-condensed ring or of a condensed ring system containing that ring
38with the nitrogen atom of at least one amino group being part of any of the groups , X being a hetero atom, Y being any atom, e.g. N-acylaminosulfones
40Y being a hydrogen or a carbon atom
C07D 295/135
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
295Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2.] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
04with substituted hydrocarbon radicals attached to ring nitrogen atoms
12substituted by singly or doubly bound nitrogen atoms
135with the ring nitrogen atoms and the substituent nitrogen atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
Applicants
  • LABORATORIOS DEL DR. ESTEVE, S. A. [ES]/[ES] (AllExceptUS)
  • SICRE GONZÁLEZ, Cristina [ES]/[ES] (UsOnly)
  • CAAMAÑO MOURE, Ana María [ES]/[ES] (UsOnly)
  • TORRENS JOVER, Antonio [ES]/[ES] (UsOnly)
Inventors
  • SICRE GONZÁLEZ, Cristina
  • CAAMAÑO MOURE, Ana María
  • TORRENS JOVER, Antonio
Agents
  • PONTI SALES, Adelaida
Priority Data
08384003.318.03.2008EP
Publication Language English (en)
Filing Language English (EN)
Designated States
Title
(EN) PROCESS FOR THE PREPARATION OF N-(1-PHENYLETHYL)ANILINES, SALTS, AND SOLVATES THEREOF USEFUL AS SEROTONIN 5-HT6 ANTAGONISTS
(FR) PROCÉDÉ POUR L'ÉLABORATION DE N-(1-PHÉNYLÉTHYL)ANILINES, DE CERTAINS DE LEURS SELS, ET SOLVATES CONVENANT COMME ANTAGONISTES DE LA SÉROTONINE (5-HT6)
Abstract
(EN) The invention relates to a process for preparing N-(1-10 phenylethyl)anilines, salts, and solvates thereof, to novel intermediates, and to the use of the intermediates in the preparation of serotonin 5-HT6 antagonists.
(FR) La présente invention concerne, d'une part un procédé pour l'élaboration de N-(1-10 phényléthyl)anilines et de certains de leurs sels et solvates, d'autre part de nouveaux intermédiaires, et enfin l'utilisation de ces intermédiaires pour l'élaboration d'antagonistes de la sérotonine (5-HT6).
Related patent documents
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