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1. (WO2009115393) PROCESS FOR THE PREPARATION OF N-(1-PHENYLETHYL)ANILINES, SALTS, AND SOLVATES THEREOF USEFUL AS SEROTONIN 5-HT6 ANTAGONISTS
Latest bibliographic data on file with the International Bureau   

Pub. No.: WO/2009/115393 International Application No.: PCT/EP2009/052066
Publication Date: 24.09.2009 International Filing Date: 20.02.2009
IPC:
C07C 211/00 (2006.01) ,C07D 295/00 (2006.01) ,C07C 251/00 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
211
Compounds containing amino groups bound to a carbon skeleton
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
295
Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
251
Compounds containing nitrogen atoms doubly- bound to a carbon skeleton
Applicants:
SICRE GONZÁLEZ, Cristina [ES/ES]; ES (UsOnly)
CAAMAÑO MOURE, Ana María [ES/ES]; ES (UsOnly)
TORRENS JOVER, Antonio [ES/ES]; ES (UsOnly)
LABORATORIOS DEL DR. ESTEVE, S. A. [ES/ES]; Av. de la Mare de Du de Montserrat, 221 E-08041 Barcelona, ES (AllExceptUS)
Inventors:
SICRE GONZÁLEZ, Cristina; ES
CAAMAÑO MOURE, Ana María; ES
TORRENS JOVER, Antonio; ES
Agent:
PONTI SALES, Adelaida; C. Consell de Cent, 322 E-08007 Barcelona, ES
Priority Data:
08384003.318.03.2008EP
Title (EN) PROCESS FOR THE PREPARATION OF N-(1-PHENYLETHYL)ANILINES, SALTS, AND SOLVATES THEREOF USEFUL AS SEROTONIN 5-HT6 ANTAGONISTS
(FR) PROCÉDÉ POUR L'ÉLABORATION DE N-(1-PHÉNYLÉTHYL)ANILINES, DE CERTAINS DE LEURS SELS, ET SOLVATES CONVENANT COMME ANTAGONISTES DE LA SÉROTONINE (5-HT6)
Abstract:
(EN) The invention relates to a process for preparing N-(1-10 phenylethyl)anilines, salts, and solvates thereof, to novel intermediates, and to the use of the intermediates in the preparation of serotonin 5-HT6 antagonists.
(FR) La présente invention concerne, d'une part un procédé pour l'élaboration de N-(1-10 phényléthyl)anilines et de certains de leurs sels et solvates, d'autre part de nouveaux intermédiaires, et enfin l'utilisation de ces intermédiaires pour l'élaboration d'antagonistes de la sérotonine (5-HT6).
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Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (EPO) (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)