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1. (WO2009059030) PYRAZOLE DERIVATIVES AS KINASE INHIBITORS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2009/059030    International Application No.:    PCT/US2008/081829
Publication Date: 07.05.2009 International Filing Date: 30.10.2008
IPC:
A01N 43/56 (2006.01)
Applicants: BURNHAM INSTITUTE FOR MEDICAL RESEARCH [US/US]; 10901 North Torrey Pines Road, La Jolla, CA 92037 (US) (For All Designated States Except US).
PELLECCHIA, Maurizio [US/US]; (US) (For US Only)
Inventors: PELLECCHIA, Maurizio; (US)
Agent: HAILE, Lisa, A.; DLA Piper LLP, 4365 Executive Drive, Suite 1100, San Diego, CA 92121-2133 (US)
Priority Data:
60/984,302 31.10.2007 US
Title (EN) PYRAZOLE DERIVATIVES AS KINASE INHIBITORS
(FR) DÉRIVÉS DE PYRAZOLE EN TANT QU'INHIBITEURS DE KINASE
Abstract: front page image
(EN)The present invention provides compounds having the general structure (I), or a pharmaceutically acceptable salt thereof wherein X is a six-member ring selected from phenyl, pyridine, or pyrimidine; Y is H, an alkenyl, a substituted alkenyl, or alkynyl, and R is H or alkyl. Pharmaceutical compositions for treating various disorders such as cancers, the compositions including compound (I) are also provided.
(FR)La présente invention concerne des composés de structure générale (I), ou un de leurs sels pharmaceutiquement acceptables, X représentant un cycle à six chaînons choisi parmi phényle, pyridine ou pyrimidine; Y représentant H, un alcényle, un alcényle substitué ou un alcynyle, et R représentant H ou un alkyle. L'invention concerne également des compositions pharmaceutiques pour le traitement de diverses maladies telles que les cancers, lesdites compositions comprenant le composé (I).
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MT, NL, NO, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)