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1. (WO2008100459) DERIVATIVES AND ANALOGS OF CHROMAN AS FUNCTIONALLY SELECTIVE ALPHA2C ADRENORECEPTOR AGONISTS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2008/100459    International Application No.:    PCT/US2008/001770
Publication Date: 21.08.2008 International Filing Date: 11.02.2008
IPC:
C07D 405/06 (2006.01), C07D 405/08 (2006.01), C07D 405/14 (2006.01), C07D 409/06 (2006.01), C07D 417/14 (2006.01), C07D 491/052 (2006.01), A61K 31/353 (2006.01), A61P 25/06 (2006.01)
Applicants: SCHERING CORPORATION [US/US]; 2000 Galloping Hill Road, Kenilworth, New Jersey 07033-0530 (US) (For All Designated States Except US).
ZHENG, Junying [CN/US]; (US) (For US Only).
MCCORMICK, Kevin, D. [US/US]; (US) (For US Only).
CHAO, Jianhua [CN/US]; (US) (For US Only).
BOYCE, Christopher, W. [US/US]; (US) (For US Only).
ASLANIAN, Robert, G. [US/US]; (US) (For US Only).
YU, Younong [CN/US]; (US) (For US Only)
Inventors: ZHENG, Junying; (US).
MCCORMICK, Kevin, D.; (US).
CHAO, Jianhua; (US).
BOYCE, Christopher, W.; (US).
ASLANIAN, Robert, G.; (US).
YU, Younong; (US)
Agent: RUSSELL, Mark, W.; Schering-Plough Corporation, Patent Department, K-6-1 1990, 2000 Galloping Hill Road, Kenilworth, New Jersey 07033-0530 (US)
Priority Data:
60/901,071 13.02.2007 US
60/972,892 17.09.2007 US
Title (EN) DERIVATIVES AND ANALOGS OF CHROMAN AS FUNCTIONALLY SELECTIVE ALPHA2C ADRENORECEPTOR AGONISTS
(FR) DÉRIVÉS ET ANALOGUES DE CHROMANE EN TANT QU'AGONISTES FONCTIONNELLEMENT SÉLECTIFS DES RÉCEPTEURS ADRÉNERGIQUES ALPHA2C
Abstract: front page image
(EN)In its many embodiments, the present invention provides a novel class of chroman compounds of formula I as α2C adrenergic receptor agonists, methods of preparing such compounds, pharmaceutical compositions containing one or more such compounds, methods of prepaxing pharmaceutical formulations comprising one or more such compounds, and methods of treatment, prevention, inhibition, or amelioration of one or more conditions associated with the α2C adrenergic receptors using such compounds or pharmaceutical compositions.
(FR)L'invention concerne, dans ses nombreux modes de réalisation, une nouvelle classe de composés chromane de formule (I) en tant qu'agonistes des récepteurs adrénergiques α2C, des procédés de préparation de ces composés, des compositions pharmaceutiques contenant un ou plusieurs de ces composés, des procédés de préparation de formulations pharmaceutiques comprenant un ou plusieurs de ces composés, ainsi que des méthodes pour le traitement, la prévention, l'inhibition ou l'amélioration d'une ou plusieurs pathologies associées aux récepteurs adrénergiques α2C à l'aide de ces composés ou compositions pharmaceutiques.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MT, NL, NO, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)