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1. WO2007149728 - ARYL AND HETEROARYL TETRAHYDROBENZAZEPINE DERIVATIVES AND THEIR USE FOR TREATING GLAUCOMA

Publication Number WO/2007/149728
Publication Date 27.12.2007
International Application No. PCT/US2007/070931
International Filing Date 12.06.2007
IPC
A61K 31/55 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
55having seven-membered rings, e.g. azelastine, pentylenetetrazole
C07D 223/16 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
223Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
14condensed with carbocyclic rings or ring systems
16Benzazepines; Hydrogenated benzazepines
A61P 27/06 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
27Drugs for disorders of the senses
02Ophthalmic agents
06Antiglaucoma agents or miotics
CPC
A61K 31/55
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
55having seven-membered rings, e.g. azelastine, pentylenetetrazole
C07D 223/16
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
223Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
14condensed with carbocyclic rings or ring systems
16Benzazepines; Hydrogenated benzazepines
Applicants
  • ALCON RESEARCH, Ltd. [US]/[US]
  • MOHAPATRA, Suchismita [IN]/[US] (UsOnly)
  • HELLBERG, Mark, R. [US]/[US] (UsOnly)
  • FENG, Zixia [US]/[US] (UsOnly)
Inventors
  • MOHAPATRA, Suchismita
  • HELLBERG, Mark, R.
  • FENG, Zixia
Agents
  • RYAN, Patrick, M.
Priority Data
60/814,97120.06.2006US
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) ARYL AND HETEROARYL TETRAHYDROBENZAZEPINE DERIVATIVES AND THEIR USE FOR TREATING GLAUCOMA
(FR) DÉRIVÉS D'ARYL ET D'HÉTÉROARYL TÉTRAHYDROBENZAZÉPINE ET LEUR UTILISATION POUR TRAITER LE GLAUCOME
Abstract
(EN)
Aryl tetrahydrobenzazepine derivatives with minimal 5-HT2B activity relative to 5-HT2A and 5-HT2C activity that are useful for treating glaucoma are disclosed.
(FR)
La présente invention concerne des dérivés d'aryl tétrahydrobenzazépine qui ont une activité 5-HT2B minimale par rapport à leurs activités 5-HT2A et 5-HT2C et qui sont utiles pour traiter le glaucome.
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