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1. WO2007138048 - NOVEL HETEROCYCLIC COMPOUNDS

Publication Number WO/2007/138048
Publication Date 06.12.2007
International Application No. PCT/EP2007/055188
International Filing Date 29.05.2007
Chapter 2 Demand Filed 31.03.2008
IPC
C07D 213/68 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
213Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
02having three double bonds between ring members or between ring members and non-ring members
04having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
60with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
62Oxygen or sulfur atoms
63One oxygen atom
68attached in position 4
A61K 31/44 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
435having six-membered rings with one nitrogen as the only ring hetero atom
44Non-condensed pyridines; Hydrogenated derivatives thereof
A61P 33/06 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
33Antiparasitic agents
02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
06Antimalarials
CPC
A61P 33/02
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
33Antiparasitic agents
02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
A61P 33/06
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
33Antiparasitic agents
02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
06Antimalarials
C07D 213/68
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
213Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
02having three double bonds between ring members or between ring members and non-ring members
04having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
60with heteroatoms or with carbon atoms having three bonds to hetero atoms, with at the most one to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
62Oxygen or sulfur atoms
63One oxygen atom
68attached in position 4
Y10S 514/895
YSECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
10TECHNICAL SUBJECTS COVERED BY FORMER USPC
STECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
514Drug, bio-affecting and body treating compositions
895Malaria
Applicants
  • GLAXO GROUP LIMITED [GB]/[GB] (AllExceptUS)
  • BUENO CALDERON, Jose Maria [ES]/[ES] (UsOnly)
  • CHICHARRO GONZALO, Jesus [ES]/[ES] (UsOnly)
  • LORENZO GARCIA, Milagros [ES]/[ES] (UsOnly)
  • MANZANO CHINCHON, M Pilar [ES]/[ES] (UsOnly)
Inventors
  • BUENO CALDERON, Jose Maria
  • CHICHARRO GONZALO, Jesus
  • LORENZO GARCIA, Milagros
  • MANZANO CHINCHON, M Pilar
Agents
  • SARDHARWALA, Fatema
Priority Data
06381025.331.05.2006EP
07380072.408.03.2007EP
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) NOVEL HETEROCYCLIC COMPOUNDS
(FR) NOUVEAUX COMPOSÉS HÉTÉROCYCLIQUES
Abstract
(EN)
4-pyridone (4-pyridinone) derivatives of Formula I and pharmaceutically acceptable derivatives thereof, processes for their preparation, pharmaceutical formulations thereof and their use in chemotherapy of certain parasitic infections such as malaria, are provided.
(FR)
L'invention concerne des dérivés de la 4-pyridone (4-pyridinone) de Formule I et des dérivés pharmaceutiquement acceptables de ceux-ci, des procédés permettant de les préparer, des formulations pharmaceutiques de ceux-ci et leur utilisation en chimiothérapie de certaines infections parasitaires, telles que la malaria.
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