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1. (WO2007125414) 9A-SUBSTITUTED AZALIDES FOR THE TRATMENT OF MALARIA
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2007/125414    International Application No.:    PCT/IB2007/001216
Publication Date: 08.11.2007 International Filing Date: 01.05.2007
Chapter 2 Demand Filed:    29.02.2008    
IPC:
A61K 31/395 (2006.01), A61K 31/7052 (2006.01), A61P 33/06 (2006.01)
Applicants: GLAXOSMITHKLINE ISTRAZIVACKI CENTAR ZAGREB D.O.O. [HR/HR]; Prilaz baruna Filipovica 29, 10000 Zagreb (HR) (For All Designated States Except US).
ALIHODZIC, Sulejman [HR/HR]; (HR) (For US Only).
FAJDETIC, Andrea [HR/HR]; (HR) (For US Only).
HUTINEC, Antun [HR/HR]; (HR) (For US Only).
IVEZIC, Zrinka [HR/HR]; (HR) (For US Only).
KUJUNDZIC, Nedjeljko [HR/HR]; (HR) (For US Only).
RUPCIC, Renata [HR/HR]; (HR) (For US Only)
Inventors: ALIHODZIC, Sulejman; (HR).
FAJDETIC, Andrea; (HR).
HUTINEC, Antun; (HR).
IVEZIC, Zrinka; (HR).
KUJUNDZIC, Nedjeljko; (HR).
RUPCIC, Renata; (HR)
Agent: CRAWLEY, Karen; GlaxoSmithKline, CIP (CN925.1), 980 Great West Road, Brentford, Middlesex TW8 9GS (GB)
Priority Data:
60/797,505 03.05.2006 US
Title (EN) 9A-SUBSTITUTED AZALIDES FOR THE TRATMENT OF MALARIA
(FR) 9A-AZALIDES SUBSTITUÉS
Abstract: front page image
(EN)The present invention relates to novel 9a-substituted azalides having antimalarial activity. More particularly, the invention relates to 9a-substituted 9a-aza-9-deoxo-9-dihydro-9a-homoerythromycin A, 3-O-decladinosyl-9a-aza-9-deoxo-9-dihydro-9a-homoerythromycin A and 3-O-decladinosyl-5-O-dedesosaminyl-9a-aza-9-deoxo-9-dihydro-9a-homoerythromycin A compounds having antimalarial activity, to the method of preparation, to the method of use, and to pharmaceutically acceptable derivatives thereof having antimalarial activity.
(FR)La présente invention concerne de nouveaux 9a-azalides substitués ayant une activité antipaludéenne. Plus précisément, l'invention concerne des composés de 9a-aza-9-deoxo-9-dihydro-9a-homoerythromycine A substituée en 9a, de 3-O-décladinosyl-9a-aza-9-deoxo-9-dihydro-9a-homoerythromycine A et de 3-O-décladinosyl-5-O-dédésosaminyl-9a-aza-9-deoxo-9-dihydro-9a-homoerytromycine A ayant une activité antipaludéenne, le procédé de préparation, le procédé d'utilisation et les dérivés pharmaceutiquement acceptables de ceux-ci ayant une activité antipaludéenne.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, MT, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)