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1. (WO2007044813) PYRIDOPYRIMIDINONE INHIBITORS OF PI3K&agr;
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2007/044813 International Application No.: PCT/US2006/039734
Publication Date: 19.04.2007 International Filing Date: 09.10.2006
IPC:
C07D 471/04 (2006.01) ,A61K 31/505 (2006.01) ,A61P 35/00 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
471
Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/-C07D463/251
02
in which the condensed system contains two hetero rings
04
Ortho-condensed systems
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
495
having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
505
Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
35
Antineoplastic agents
Applicants:
EXELIXIS, INC. [US/US]; 210 East Grand Avenue, P.O. Box 511 South San Francisco, CA 94083-0511, US (AllExceptUS)
BAIK, Tae-Gon [KR/US]; US (UsOnly)
BUHR, Chris, A. [US/US]; US (UsOnly)
LARA, Katherine [US/US]; US (UsOnly)
MA, Sunghoon [KR/US]; US (UsOnly)
MAC, Morrison [US/US]; US (UsOnly)
NUSS, John, M. [US/US]; US (UsOnly)
WANG, Longcheng [CN/US]; US (UsOnly)
WANG, Yong [CN/US]; US (UsOnly)
YEUNG, Bryan, K. S. [SG/SG]; SG (UsOnly)
Inventors:
BAIK, Tae-Gon; US
BUHR, Chris, A.; US
LARA, Katherine; US
MA, Sunghoon; US
MAC, Morrison; US
NUSS, John, M.; US
WANG, Longcheng; US
WANG, Yong; US
YEUNG, Bryan, K. S.; SG
Agent:
WADE, Janice, V. ; Exelixis, INC 210 East Grand Avenue P.O. Box 511 South San Francisco, CA 94083-0511, US
Priority Data:
60/724,57107.10.2005US
60/743,71923.03.2006US
Title (EN) PYRIDOPYRIMIDINONE INHIBITORS OF PI3K&agr;
(FR) INHIBITEURS DE PI3K&agr; DE TYPE PYRIDOPYRIMIDINONE
Abstract:
(EN) The invention is directed to Compounds of Formula (I) and pharmaceutically acceptable salts or solvates thereof, as well as methods of making and using the compounds.
(FR) La présente invention porte sur des Composés de Formule (I) ainsi que sur les sels ou les solvates de qualité pharmaceutique desdits composés, de même que sur les méthodes de synthèse et d'utilisation desdits composés.
front page image
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LV, LY, MA, MD, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, SV, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)
Also published as:
NO20082090RSP-2013/0400UAa200804287MXMX/a/2008/004401KR1020080056195IL190292
EP1940839EP2322523ZA2008/02585JP2009511504US20090270430CN101395155
CA2623770EA200800760ES2432046BRPI0617159KR1020130140145KR1020140105621
NZ566903AU2006302078DK1940839IN1169/KOLNP/2008