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Machine translation
1. (WO2007010082) PROCESS FOR PREPARING A 3-ARYLOXY-3-ARYLPROPYLAMINE
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2007/010082    International Application No.:    PCT/FI2006/000252
Publication Date: 25.01.2007 International Filing Date: 14.07.2006
IPC:
C07C 213/06 (2006.01), C07C 217/48 (2006.01)
Applicants: FERMION OY [FI/FI]; Koivu-Mankkaan tie 6 A, FI-02200 Espoo (FI) (For All Designated States Except US).
GRUMANN, Arne [DE/FI]; (FI) (For US Only).
LAPPALAINEN, Kari [FI/FI]; (FI) (For US Only).
MAIWALD, Peter [DE/FI]; (FI) (For US Only).
PIETIKÄINEN, Pekka [FI/FI]; (FI) (For US Only).
RUMMAKKO, Petteri [FI/FI]; (FI) (For US Only)
Inventors: GRUMANN, Arne; (FI).
LAPPALAINEN, Kari; (FI).
MAIWALD, Peter; (FI).
PIETIKÄINEN, Pekka; (FI).
RUMMAKKO, Petteri; (FI)
Agent: ORION CORPORATION ORION PHARMA; Legal Affairs and Intellectual Property Rights, P.O. Box 65, FI-02101 Espoo (FI)
Priority Data:
60/699,502 15.07.2005 US
20055413 15.07.2005 FI
Title (EN) PROCESS FOR PREPARING A 3-ARYLOXY-3-ARYLPROPYLAMINE
(FR) PROCEDE D'ELABORATION DE COMPOSE
Abstract: front page image
(EN)The invention relates to the use of copper-catalyzed nucleophilic aromatic substitution reaction for preparing 3-aryloxy-3-arylpropylamines and more specifically to a method of preparing certain 3-aryloxy-3-arylpropylamines and the pharmaceutically acceptable addition salts thereof, comprising reacting an amino alcohol with a haloaromatic compound in the presence of a base and a catalytic copper source, and in the absence of a separate ligand.
(FR)Utilisation de réaction de substitution aromatique nucléophile catalysée au cuivre pour l'élaboration de 3-aryloxy-3-arylpropylamines et plus précisément procédés d'élaboration de certaines 3-aryloxy-3-arylpropylamines y compris leurs sels d'addition pharmaceutiquement acceptables, par réaction entre amino alcool et composé halo-aromatique en présence d'une base et d'une source de cuivre catalytique, et en l'absence de ligand séparé.
Designated States: AE, AG, AL, AM, AT, AU, AZ, BA, BB, BG, BR, BW, BY, BZ, CA, CH, CN, CO, CR, CU, CZ, DE, DK, DM, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LV, LY, MA, MD, MG, MK, MN, MW, MX, MZ, NA, NG, NI, NO, NZ, OM, PG, PH, PL, PT, RO, RS, RU, SC, SD, SE, SG, SK, SL, SM, SY, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LS, MW, MZ, NA, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)